Report error Found 1715 with Last Name = 'monga' and Initial = 'v'
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 4.90nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
Affinity DataKd: 4.80E+3nMAssay Description:Binding affinity to DNA-tagged Aurora B (unknown origin) expressed in mammalian system assessed as binding constant (Kd) by competition binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 67nMAssay Description:Binding affinity to DNA-tagged EGFR (unknown origin) expressed in bacterial system assessed as binding constant (Kd) by competition binding assayMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Rat)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Agonist activity at TRHR2 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
Affinity DataKd: 3.40E+3nMAssay Description:Binding affinity to DNA-tagged Aurora A (unknown origin) expressed in mammalian system assessed as binding constant (Kd) by competition binding assayMore data for this Ligand-Target Pair
TargetThyrotropin-releasing hormone receptor(Human)
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
National Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at TRHR1 expressed in HEK293EM cells assessed as activation potency by measuring CREB-luciferase reporter activityMore data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.460nMAssay Description:Inhibition of Aurora A (unknown origin) using kemptide as substrate incubated for 50 mins in the presence of ATP by ADP-Glo reagent based luminescenc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inverse agonist activity at human A2A receptor assessed as inhibition of cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inverse agonist activity at human A2A receptor assessed as inhibition of basal cAMP levelMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Inverse agonist activity at human A2A receptor assessed as inhibition of cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant sEHMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1 by spectrophotometer based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1 by spectrophotometer based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1 by spectrophotometer based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1More data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1 by spectrophotometer based analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human CA1More data for this Ligand-Target Pair




























