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TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at PPARgamma (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508101(CHEMBL4521388)
Affinity DataEC50:  1.66E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508102(CHEMBL4537335)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508103(CHEMBL4589453)
Affinity DataEC50:  2.25E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508104(CHEMBL4591405)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508105(CHEMBL4542891)
Affinity DataEC50:  730nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508106(CHEMBL4517263)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508107(CHEMBL4574542)
Affinity DataEC50:  1.09E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508108(CHEMBL4567211)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508109(CHEMBL4592935)
Affinity DataEC50:  1.03E+4nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataEC50:  460nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508113(CHEMBL4453360)
Affinity DataEC50:  2.72E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508114(CHEMBL4466241)
Affinity DataEC50:  1.32E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508115(CHEMBL4469751)
Affinity DataEC50:  1.81E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508116(CHEMBL4535401)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508117(CHEMBL4463602)
Affinity DataEC50:  2.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508118(CHEMBL4436393)
Affinity DataEC50:  7.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508119(CHEMBL4472191)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508120(CHEMBL4531918)
Affinity DataEC50:  2.62E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508121(CHEMBL4527893)
Affinity DataEC50:  2.36E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508122(CHEMBL4456647)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508123(CHEMBL4452865)
Affinity DataEC50:  3.31E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508112(CHEMBL4546437)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508124(CHEMBL4443588)
Affinity DataEC50:  1.53E+3nMAssay Description:Agonist activity at human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467129(CHEMBL4278280)
Affinity DataIC50: 0.700nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557417(CHEMBL4762591)
Affinity DataIC50: 1nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557413(CHEMBL4758377)
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557417(CHEMBL4762591)
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557433(CHEMBL4746891)
Affinity DataIC50: 1nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467130(CHEMBL4291216)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508111(CHEMBL4520827)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467140(CHEMBL4289788)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467133(CHEMBL4280574)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467135(CHEMBL4287379)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557416(CHEMBL4786982)
Affinity DataIC50: 2nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557396(CHEMBL4747683)
Affinity DataIC50: 2nMAssay Description:Inhibition of DPP4 (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467138(CHEMBL4282931)
Affinity DataIC50: 2.10nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467131(CHEMBL4288964)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50508110(CHEMBL4444760)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50009366(CHEMBL3233842 | US9346814, Cmpd No 1, Example 1 | ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557415(CHEMBL4750058)
Affinity DataIC50: 4nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364573(CHEMBL1951143)
Affinity DataIC50: 4.5nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467139(CHEMBL4293170)
Affinity DataIC50: 4.70nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557434(CHEMBL4780357)
Affinity DataIC50: 5nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557439(CHEMBL4758299)
Affinity DataIC50: 5nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetProlyl endopeptidase(Human)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557414(CHEMBL4748328)
Affinity DataIC50: 5nMAssay Description:Inhibition of PREP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor(Human)
Boryung Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50467136(CHEMBL4284022)
Affinity DataIC50: 5.60nMAssay Description:Antagonist activity at type-1 angiotensin 2 receptor (unknown origin) by calcium mobilizing assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557442(CHEMBL4747575)
Affinity DataIC50: 7nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetAcyl-protein thioesterase 1(Rat)
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM50557438(CHEMBL4789965)
Affinity DataIC50: 9nMAssay Description:Inhibition of FAP (unknown origin) using AMC substrate by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
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