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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614556(US20230270751, Example 127 | (5S)-2-(6- Ethylpyrid...)
Affinity DataEC50:  41nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614618(US20230270751, Example 110-1 | (6R*)-N-[(3S)-9- fl...)
Affinity DataEC50:  42nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetTyrosine-protein kinase HCK(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  5nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), were evaluated in a similar fashion to that descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614577(US20230270751, Example 148 | N-[(3S)-9-fluoro-2- o...)
Affinity DataEC50:  72nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetMitogen-activated protein kinase 12(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  5nMAssay Description:The inhibitory activities of compounds of the invention against p38MAPKγ (MAPK12: Invitrogen), were evaluated in a similar fashion to that descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2019
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614631(US20230270751, Example 191-2 | (5S*)-N-[(3S)-9- fl...)
Affinity DataEC50:  280nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614449(US20230270751, Example 26 | (5S)-2-(2- Fluoropheny...)
Affinity DataEC50:  43nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetTyrosine-protein kinase SYK(Human)
Respivert

US Patent
LigandPNGBDBM161376(US9108950, 1 | US9724347, Example 1 | US10238658, ...)
Affinity DataKd:  14nMAssay Description:The kinase enzyme binding activities of compounds disclosed herein were determined using a proprietary assay which measures active site-directed comp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/18/2016
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614572(US20230270751, Example 143 | 2-[2-Fluoro-4- (methy...)
Affinity DataEC50:  149nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614495(US20230270751, Example 72 | (5R)-2-(2-Fluoro-6- me...)
Affinity DataEC50:  100nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614542(US20230270751, Example 113 | N-[(3S)-9-fluoro-2- o...)
Affinity DataEC50:  53nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetGlycogen synthase kinase-3 alpha(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  180nMAssay Description:The GSK3-α protein (500 ng/mL, 2.5 μL) was mixed with the test compound (2.5 μL at either 4 μg/mL, 0.4 μg/mL, 0.04 μg/m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2019
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614602(US20230270751, Example 172 | N-[(3S)-9-fluoro-2- o...)
Affinity DataEC50:  235nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetMitogen-activated protein kinase 14(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  1nMAssay Description:p38 MAPKα: The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), were evaluated indirectly by det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2021
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614567(US20230270751, Example 138 | 2-(4-Cyano-2- fluorop...)
Affinity DataEC50:  54nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614570(US20230270751, Example 141 | (5R)-2-(2-Fluoro-4- m...)
Affinity DataEC50:  20nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614595(US20230270751, Example 166 | 5- [(Dimethylamino)me...)
Affinity DataEC50:  201nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614540(US20230270751, Example 111 | (5R)-N-[(3S)-9- fluor...)
Affinity DataEC50:  64nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614439(US20230270751, Example 16 | N-[(3S)-2-Oxo-5- pheny...)
Affinity DataEC50:  454nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614453(US20230270751, Example 30 | (5R)-N-[(3S)-9- fluoro...)
Affinity DataEC50:  16nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614522(US20230270751, Example 99 | 2-(1-Ethylpyrazol-4- y...)
Affinity DataEC50:  71nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614578(US20230270751, Example 149 | 2-(1-Methylindazol- 4...)
Affinity DataEC50:  194nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614508(US20230270751, Example 85 | (5R)-2-[6-(2-Hydroxy-2...)
Affinity DataEC50:  121nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614551(US20230270751, Example 122 | (5R)-N-[(3S)-9- fluor...)
Affinity DataEC50:  166nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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Target5-hydroxytryptamine receptor 2A(Human)
Respivert

US Patent
LigandPNGBDBM161376(US9108950, 1 | US9724347, Example 1 | US10238658, ...)
Affinity DataKd:  20nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), were evaluated indirectly by determining the lev...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2019
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614580(US20230270751, Example 151 | N-[(3S)-2-oxo-5- phen...)
Affinity DataEC50:  108nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614474(US20230270751, Example 51 | (5R)-2-(3- Fluoropyrid...)
Affinity DataEC50:  80nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetMitogen-activated protein kinase 14(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), were evaluated indirectly by determining the lev...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 12(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  5nMAssay Description:The inhibitory activities of compounds of the invention against p38MAPKγ (MAPK12: Invitrogen), were evaluated in a similar fashion to that descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614605(US20230270751, Example 175 | 2-(2-Fluorophenyl)- 6...)
Affinity DataEC50:  61nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614426(US20230270751, Example 3 | 2-[6-(Ethylamino)-2- fl...)
Affinity DataEC50:  20nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614488(US20230270751, Example 65 | (5R)-2-(6-Ethyl-2- met...)
Affinity DataEC50:  84nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614596(US20230270751, Example 167 | N-[(3S)-9-fluoro-2- o...)
Affinity DataEC50:  91nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
Respivert

US Patent
LigandPNGBDBM161376(US9108950, 1 | US9724347, Example 1 | US10238658, ...)
Affinity DataKd:  10nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), were evaluated in a similar fashion to that descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2019
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614481(US20230270751, Example 58 | (5R)-2-(2,6-Dimethyl- ...)
Affinity DataEC50:  188nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614600(US20230270751, Example 171 | US20230270751, Exampl...)
Affinity DataEC50:  59nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Respivert

US Patent
LigandPNGBDBM161376(US9108950, 1 | US9724347, Example 1 | US10238658, ...)
Affinity DataKd:  1.20E+3nMAssay Description:The GSK3-α protein (500 ng/mL, 2.5 μL) was mixed with the test compound (2.5 μL at either 4 μg/mL, 0.4 μg/mL, 0.04 μg/m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2019
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614642(US20230270751, Example 202 | (2R)-6-(2- Fluorophen...)
Affinity DataEC50:  127nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614590(US20230270751, Example 161 | (5R)-N-[(3S)-9- fluor...)
Affinity DataEC50:  54nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614630(US20230270751, Example 191-1 | (5R*)-N-[(3S)-9- fl...)
Affinity DataEC50:  83nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614530(US20230270751, Example 106 | US20230270751, Exampl...)
Affinity DataEC50:  66nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614613(US20230270751, Example 183 | (5R)-N-[(3S)-9- fluor...)
Affinity DataEC50:  294nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614507(US20230270751, Example 84 | (5R)-2-(1-Ethylpyrazol...)
Affinity DataEC50:  70nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614537(US20230270751, Example 108 | tert-butyl N-ethyl-N-...)
Affinity DataEC50:  117nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614457(US20230270751, Example 34 | 2-(2,4- Difluorophenyl...)
Affinity DataEC50:  143nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614490(US20230270751, Example 67 | (5R)-N-[(3S)-9-fluoro-...)
Affinity DataEC50:  19nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614573(US20230270751, Example 144 | (5R)-N-[(3S)-9- fluor...)
Affinity DataEC50:  101nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614463(US20230270751, Example 40 | 2-(2-Fluorophenyl)- 6,...)
Affinity DataEC50:  57nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

TargetTyrosine-protein kinase SYK(Human)
Respivert

US Patent
LigandPNGBDBM142598(US8933228, Ref 2 | US9249125, Reference Compound |...)
Affinity DataKd:  9nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), were evaluated in a similar fashion to that descr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2019
Entry Details
Go to US Patent

TargetNucleoprotein(Human respiratory syncytial virus A (strain A2))
Reviral

US Patent
LigandPNGBDBM614550(US20230270751, Example 121 | (5R)-2-(1,5- Dimethyl...)
Affinity DataEC50:  374nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
Go to US Patent

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