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TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525018(CHEMBL4465842)
Affinity DataIC50: 440nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525017(CHEMBL4462117)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525014(CHEMBL4475419)
Affinity DataIC50: 1.73E+4nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525016(CHEMBL4457217)
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525019(CHEMBL4471561)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525020(CHEMBL4518572)
Affinity DataIC50: 3.07E+4nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetLysosomal alpha-mannosidase(Human)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525015(CHEMBL4435118)
Affinity DataIC50: 1.16E+5nMAssay Description:Inhibition of Lysosomal alpha-mannosidase in wild-type human fibroblast cell lysates using 4-methylumbelliferone alpha-D-mannopyranoside as a reporte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222179(m-tolyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbo...)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222191(2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222188(phenyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbox...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222183(o-tolyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbo...)
Affinity DataKi:  220nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  300nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222178(thiophen-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopen...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525015(CHEMBL4435118)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525016(CHEMBL4457217)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525014(CHEMBL4475419)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525017(CHEMBL4462117)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525018(CHEMBL4465842)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525020(CHEMBL4518572)
Affinity DataKi:  500nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222186(2-fluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-en...)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222185(2-(3,4-dichlorophenyl)-N-methoxycyclopent-1-enecar...)
Affinity DataKi:  830nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(furan-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopent-1...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50211023(methyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbox...)
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222176(isopropyl 2-(3,4-dichlorophenyl)cyclopent-1-enecar...)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525019(CHEMBL4471561)
Affinity DataKi:  3.20E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222177(2,2,2-trifluoroethyl 2-(3,4-dichlorophenyl)cyclope...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222186(2-fluoroethyl 2-(3,4-dichlorophenyl)cyclopent-1-en...)
Affinity DataKi:  5.80E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222192(2-(3,4-dichlorophenyl)-N-methoxy-N-methylcyclopent...)
Affinity DataKi:  6.40E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-mannosidase(Jack bean)
University of Sevilla

Curated by ChEMBL
LigandPNGBDBM50525021(CHEMBL4483772)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of jack bean Lysosomal alpha-mannosidase assessed as residual hydrolytic activity after 10 to 30 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222191(2-(3,4-dichlorophenyl)-N-(2-fluoroethyl)cyclopent-...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222189(N-cyclobutyl-2-(3,4-dichlorophenyl)cyclopent-1-ene...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222185(2-(3,4-dichlorophenyl)-N-methoxycyclopent-1-enecar...)
Affinity DataKi:  9.20E+3nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222180((2-(3,4-dichlorophenyl)cyclopent-1-enyl)(morpholin...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50211023(methyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbox...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222190(cyclohexyl 2-(3,4-dichlorophenyl)cyclopent-1-eneca...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222184(2-(3,4-dichlorophenyl)-N-(thiophen-2-ylmethyl)cycl...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(furan-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopent-1...)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222175(2-(3,4-dichlorophenyl)-N-(furan-2-ylmethyl)cyclope...)
Affinity DataKi:  2.40E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222176(isopropyl 2-(3,4-dichlorophenyl)cyclopent-1-enecar...)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222183(o-tolyl 2-(3,4-dichlorophenyl)cyclopent-1-enecarbo...)
Affinity DataKi:  3.30E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222178(thiophen-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopen...)
Affinity DataKi:  4.20E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetBeta-glucosidase(Cherry)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50186735(D-1,4-dideoxy-4,4-difluoromannonojirimycin | CHEMB...)
Affinity DataKi:  4.50E+4nMpH: 6.8Assay Description:Inhibition of almond beta glucosidase at pH 6.8More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222182(2-hydroxyethyl 2-(3,4-dichlorophenyl)cyclopent-1-e...)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human SERT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222189(N-cyclobutyl-2-(3,4-dichlorophenyl)cyclopent-1-ene...)
Affinity DataKi:  5.00E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222181((2-(3,4-dichlorophenyl)cyclopent-1-enyl)(pyrrolidi...)
Affinity DataKi:  5.80E+4nMAssay Description:Displacement of [125I]RTI55 from human DAT transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent noradrenaline transporter(Human)
University of Aarhus

Curated by ChEMBL
LigandPNGBDBM50222187(furan-2-ylmethyl 2-(3,4-dichlorophenyl)cyclopent-1...)
Affinity DataKi:  6.10E+4nMAssay Description:Displacement of [125I]RTI55 from human NET transfected in COS1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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