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TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538690(CHEMBL4645309)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50527781(CHEMBL4456676)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538687(CHEMBL4637120)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538689(CHEMBL4640511)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetRetinal dehydrogenase 2(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataIC50: 2.76E+4nMAssay Description:Inhibition of human recombinant ALDH1A2 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetRetinal dehydrogenase 2(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538686(CHEMBL4640253)
Affinity DataIC50: 6.14E+4nMAssay Description:Inhibition of human recombinant ALDH1A2 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538686(CHEMBL4640253)
Affinity DataIC50: 8.06E+4nMAssay Description:Inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase 1A1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of human recombinant ALDH1A1 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataKi:  120nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetRetinal dehydrogenase 2(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataKi:  920nMAssay Description:Competitive inhibition of human recombinant ALDH1A2 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase family 1 member A3(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataKi:  8.70E+3nMAssay Description:Competitive inhibition of human recombinant ALDH1A3 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetRetinal dehydrogenase 2(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataKi:  2.76E+4nMAssay Description:Competitive inhibition of human recombinant ALDH1A2 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase 1A1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538688(CHEMBL4642789)
Affinity DataKi:  7.95E+4nMAssay Description:Competitive inhibition of human recombinant ALDH1A1 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetAldehyde dehydrogenase 1A1(Human)
University of Pisa

Curated by ChEMBL
LigandPNGBDBM50538685(CHEMBL4644541)
Affinity DataKi:  1.68E+5nMAssay Description:Competitive inhibition of human recombinant ALDH1A1 pre-incubated for 5 mins before acetaldehyde addition by continuous spectrometric assay relative ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed