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TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215110((1R,3R,4R,7S)-(7-hydroxy-3-(N6-(3-iodobenzyl)-aden...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataEC50:  2.40E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215115(N6-(3-Iodobenzyl)-2'-O-methyladenosine | CHEMBL428...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215119(2'-O-methyladenosine-N-methyl-5'-uronamide | CHEMB...)
Affinity DataEC50:  453nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50144945(CHEMBL73237 | (2R,3R,4R,5R)-5-(6-amino-9H-purin-9-...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215117((1S,3R,4R,7S)-3-(6-amino-purin-9-yl)-1-hydroxymeth...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215115(N6-(3-Iodobenzyl)-2'-O-methyladenosine | CHEMBL428...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215116(N6-(3-iodobenzyl)-2'-O-methyladenosine-N-methyl-5'...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215111((1S,3R,4R,7S)-7-hydroxy-1-hydroxymethyl-3-(N6-(3-i...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215118((1S,3R,4R,7S)-7-hydroxy-1-hydroxymethyl-3-(N6-(3-i...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596260(CHEMBL5183506)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215114((1R,3R,4R,7S)-(7-hydroxy-3-(adenin-9-yl)-2,5-dioxa...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215112((1R,3R,4R,7S)-3-(6-amino-purin-9-yl)-1-hydroxymeth...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50144945(CHEMBL73237 | (2R,3R,4R,5R)-5-(6-amino-9H-purin-9-...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215113((1R,3R,4R,7S)-(7-hydroxy-3-(N6-(3-iodobenzyl)-aden...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215110((1R,3R,4R,7S)-(7-hydroxy-3-(N6-(3-iodobenzyl)-aden...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215116(N6-(3-iodobenzyl)-2'-O-methyladenosine-N-methyl-5'...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215109((1R,3R,4R,7S)-(7-hydroxy-3-(adenin-9-yl)-2-oxa-5-a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215111((1S,3R,4R,7S)-7-hydroxy-1-hydroxymethyl-3-(N6-(3-i...)
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at human adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596273(CHEMBL5185133)
Affinity DataEC50:  2.50E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596262(CHEMBL5176331)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596263(CHEMBL5207657)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596264(CHEMBL5206355)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596265(CHEMBL5178897)
Affinity DataEC50:  2.60E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596266(CHEMBL5205450)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596267(CHEMBL5172698)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596268(CHEMBL5203592)
Affinity DataEC50:  500nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596269(CHEMBL5183842)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596270(CHEMBL5186572)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596271(CHEMBL5176046)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataEC50:  2.50E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596272(CHEMBL5199813)
Affinity DataEC50:  3.80E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596277(CHEMBL5198009)
Affinity DataEC50: <3.00E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596275(CHEMBL5176348)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596276(CHEMBL5207002)
Affinity DataEC50:  7.00E+3nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596274(CHEMBL5204986)
Affinity DataEC50:  8.70E+4nMAssay Description:Inhibition of hERG by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215115(N6-(3-Iodobenzyl)-2'-O-methyladenosine | CHEMBL428...)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215111((1S,3R,4R,7S)-7-hydroxy-1-hydroxymethyl-3-(N6-(3-i...)
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215110((1R,3R,4R,7S)-(7-hydroxy-3-(N6-(3-iodobenzyl)-aden...)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50144945(CHEMBL73237 | (2R,3R,4R,5R)-5-(6-amino-9H-purin-9-...)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215118((1S,3R,4R,7S)-7-hydroxy-1-hydroxymethyl-3-(N6-(3-i...)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Santaris Pharma

Curated by ChEMBL
LigandPNGBDBM50215109((1R,3R,4R,7S)-(7-hydroxy-3-(adenin-9-yl)-2-oxa-5-a...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human adenosine A3 receptor after 15 to 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596272(CHEMBL5199813)
Affinity DataIC50: 190nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM21690(Ciprinol | 1-cyclopropyl-6-fluoro-4-oxo-7-(piperaz...)
Affinity DataIC50: 230nMAssay Description:Inhibition of Escherichia coli DNA gyrase by fluorescence based microtiter plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596263(CHEMBL5207657)
Affinity DataIC50: 280nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596278(CHEMBL5178214)
Affinity DataIC50: 280nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50393503(CHEMBL2158050)
Affinity DataIC50: 340nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596275(CHEMBL5176348)
Affinity DataIC50: 370nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50596261(CHEMBL5176134)
Affinity DataIC50: 370nMAssay Description:Inhibition of Staphylococcus aureus DNA gyrase supercoiling activity using pNO1 plasmid DNA as substrate incubated for 30 mins by fluorescence based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
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