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TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Montana

Curated by ChEMBL
LigandPNGBDBM50067499((6aR,10aR)-3(1,1-dimethylheptyl)-9-hydroxymethyl)-...)
Affinity DataKi:  2.66nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418901(CHEMBL1808415)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418893(CHEMBL1808400)
Affinity DataKi:  275nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418884(CHEMBL1808414)
Affinity DataKi:  347nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University of Montana

Curated by ChEMBL
LigandPNGBDBM50354474(CHEMBL1836868)
Affinity DataKi:  387nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418896(CHEMBL1807152)
Affinity DataKi:  467nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418896(CHEMBL1807152)
Affinity DataKi:  468nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418891(CHEMBL1808405)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418898(CHEMBL1808398)
Affinity DataKi:  676nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418878(CHEMBL1808418)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418894(CHEMBL1808399)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418897(CHEMBL1808402)
Affinity DataKi:  1.07E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418892(CHEMBL1808403)
Affinity DataKi:  1.45E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418904(CHEMBL1808401)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418880(CHEMBL1808416)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418880(CHEMBL1808416)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418880(CHEMBL1808416)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418881(CHEMBL1808422)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418887(CHEMBL1808410)
Affinity DataKi:  2.04E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418879(CHEMBL1808417)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418879(CHEMBL1808417)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418878(CHEMBL1808418)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418878(CHEMBL1808418)
Affinity DataKi:  2.57E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418896(CHEMBL1807152)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418879(CHEMBL1808417)
Affinity DataKi:  3.09E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418883(CHEMBL1808420)
Affinity DataKi:  3.24E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418886(CHEMBL1808411)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Francisella tularensis subsp. tularensis (strain S...)
Naval Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50436715(CHEMBL2398661)
Affinity DataKi:  3.40E+3nMAssay Description:Competitive inhibition of C-terminal His6-tagged Francisella tularensis SCHU S4 FabI expressed in Escherichia coli BL21 (DE3) using CrCoA as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418899(CHEMBL1808413)
Affinity DataKi:  4.07E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418889(CHEMBL1808407)
Affinity DataKi:  5.13E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418888(CHEMBL1808408)
Affinity DataKi:  5.13E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418890(CHEMBL1806517)
Affinity DataKi:  6.61E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEnoyl-[acyl-carrier-protein] reductase [NADH](Francisella tularensis subsp. tularensis (strain S...)
Naval Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50436718(CHEMBL1341978)
Affinity DataKi:  7.00E+3nMAssay Description:Competitive inhibition of C-terminal His6-tagged Francisella tularensis SCHU S4 FabI expressed in Escherichia coli BL21 (DE3) using CrCoA as substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418902(CHEMBL1808409)
Affinity DataKi:  8.32E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418900(CHEMBL1808419)
Affinity DataKi:  9.55E+3nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418903(CHEMBL1808406)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418895(CHEMBL1808404)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418885(CHEMBL1808412)
Affinity DataKi:  1.74E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50418882(CHEMBL1808421)
Affinity DataKi:  2.04E+4nMAssay Description:Displacement of [3H]CCK8 from rat pancreas CCK1 receptor at by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50505991(CHEMBL4470113)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265958(CHEMBL4086507)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50505989(CHEMBL4551714)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50505994(CHEMBL4440109)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50094465(CHEMBL3590106 | US10525036, Example BVD-523 | US10...)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50505988(CHEMBL4482864)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50094464(CHEMBL3590107 | US10525036, Example SCH772984 | US...)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using Erktide as substrate preincubated with enzyme for 20 mins prior to substrate addition by...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265960(CHEMBL4098608)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 60 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50505993(CHEMBL4587118)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of MEK U911-activated ERK2 (unknown origin) using ERKtide as substrate preincubated for 20 mins followed by substrate addition in presence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50265961(CHEMBL4090886)
Affinity DataIC50: <0.300nMAssay Description:Inhibition of ERK2 (unknown origin) in the presence of 60 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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