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TargetEpithelial discoidin domain-containing receptor 1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  31nMAssay Description:Inhibition of wild-type human partial length DDR1 (R565 to V876 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 14(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  6.30nMAssay Description:Inhibition of wild-type human full length p38-alpha (M1 to S360 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMitogen-activated protein kinase 11(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  20nMAssay Description:Inhibition of wild-type human full length p38-beta (M1 to Q364 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  130nMAssay Description:Inhibition of wild-type human non-phosphorylated ABL1 (S229 to K512 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 20(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  120nMAssay Description:Inhibition of wild-type human partial length ZAK (M1 to L331 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetDiscoidin domain-containing receptor 2(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50556597(CHEMBL4756586)
Affinity DataKd:  40nMAssay Description:Inhibition of wild-type human partial length DDR2 (V555 to E855 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
LigandPNGBDBM246383(US9446044, 69)
Affinity DataKd:  7.30nMAssay Description:Binding affinity to DYRK1A (unknown origin) assessed as dissociation constant at 3 uM by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to DYRK1A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to DYRK1B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd: <100nMAssay Description:Binding affinity to CLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to CLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-3(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to PIM3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform gamma-2(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to CSNK1G2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform gamma-3(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to CSNK1G3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to CSNK1D (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to CSNK1E (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 19(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  100nMAssay Description:Binding affinity to MAP3K19 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  75nMAssay Description:Inhibition of CLK1 (H148 to I484 residues) (unknown origin) at 15 uM by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50560703(CHEMBL1349996)
Affinity DataKd:  7.78E+3nMAssay Description:Inhibition of CLK3 (R134 to T484 residues) (unknown origin) at 15 uM by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  4.60nMAssay Description:Binding affinity to human CASK by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase I isoform epsilon(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  770nMAssay Description:Binding affinity to human CSNK1E by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  570nMAssay Description:Binding affinity to human MERTK by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  740nMAssay Description:Binding affinity to human non-phosphorylated ABL1 by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-2(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to human N-terminal RSK3 kinase domain 1 by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 2(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  690nMAssay Description:Binding affinity to human MAP3K2 by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  800nMAssay Description:Binding affinity to human MET by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to human AXL by KINOMEscan scanMAX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425829(CHEMBL2312304)
Affinity DataKd:  87nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50425830(CHEMBL2312303)
Affinity DataKd:  140nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574221(CHEMBL4847568)
Affinity DataKd:  220nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574222(CHEMBL4856516)
Affinity DataKd:  630nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574223(CHEMBL4846209)
Affinity DataKd:  60nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574224(CHEMBL4876584)
Affinity DataKd:  38nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeripheral plasma membrane protein CASK(Human)
Goethe University Frankfurt Am Main

Curated by ChEMBL
LigandPNGBDBM50574225(CHEMBL4850857)
Affinity DataKd:  22nMAssay Description:Binding affinity to recombinant N-terminal His-tagged CASK (1 to 337 residues) (unknown origin) expressed in Escherichia coli assessed as dissociatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50226181(Carbamic acid 5-hydroxy-6-{4-hydroxy-3-[4-hydroxy-...)
Affinity DataKd:  7.50E+3nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575781(CHEMBL4851364)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575782(CHEMBL4873913)
Affinity DataKd:  1.42E+4nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575783(CHEMBL4871486)
Affinity DataKd:  1.57E+4nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575784(CHEMBL4845679)
Affinity DataKd:  2.75E+4nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3A(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575785(CHEMBL4851932)
Affinity DataKd:  1.72E+4nMAssay Description:Binding affinity to human LC3A expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50226181(Carbamic acid 5-hydroxy-6-{4-hydroxy-3-[4-hydroxy-...)
Affinity DataKd:  1.74E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575781(CHEMBL4851364)
Affinity DataKd:  1.14E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575782(CHEMBL4873913)
Affinity DataKd:  2.16E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575783(CHEMBL4871486)
Affinity DataKd:  2.35E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575784(CHEMBL4845679)
Affinity DataKd:  2.05E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetMicrotubule-associated proteins 1A/1B light chain 3B(Human)
Goethe-University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50575785(CHEMBL4851932)
Affinity DataKd:  2.58E+4nMAssay Description:Binding affinity to human LC3B expressed in Escherichia coli BL21-(DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetFocal adhesion kinase 1(Human)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50440378(CHEMBL2425111)
Affinity DataEC50:  3.01E+5nMAssay Description:Inhibition of N-terminal NanoLuc-tagged full length FAK (unknown origin) transfected in HEK293T cells pre-incubated with compound for 2 hrs followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
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