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TargetChaperonin GroEL(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50179360(CHEMBL3040216)
Affinity DataKd:  9.80E+3nMAssay Description:Binding affinity to Escherichia coli GroEL expressed in Escherichia coliDH5alpha by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHeat shock-related 70 kDa protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA2 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 6(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA6 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  334nMAssay Description:Binding affinity to HspA5 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataKd:  149nMAssay Description:Binding affinity to 6His-tagged BRD3-BD2 (unknown origin) by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetEukaryotic initiation factor 4A-I(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50610971(CHEMBL5290937)
Affinity DataEC50:  2.75E+4nMAssay Description:Inhibition of human recombinant N-terminal His6-tagged eIF4A expressed in Escherichia coli BL21 CodonPlus cells using ATP and yeast RNA as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataKd:  14nMAssay Description:Binding affinity to 6His-tagged BRD3-BD1 (unknown origin) by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetStress-70 protein, mitochondrial(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  7.48E+3nMAssay Description:Binding affinity to HspA9 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock cognate 71 kDa protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA8 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1A(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1A (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetHeat shock 70 kDa protein 1-like(Homo sapiens)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to HspA1L (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to human partial length BRD4 BD2 (K333 to E460 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 5.5nMAssay Description:Binding affinity to human partial length BRDT BD2 (K250 to E382 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 7.10nMAssay Description:Binding affinity to human partial length BRD3 BD1 (P24 to E144 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 7.60nMAssay Description:Binding affinity to human partial length BRD3 BD2 (G306 to P416 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 9.30nMAssay Description:Binding affinity to human partial length BRD2 BD2 (E348to D455 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 18nMAssay Description:Binding affinity to human partial length BRD4 BD1 (N44 to E168 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50: 18nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114395(CHEMBL3605564)
Affinity DataIC50: 19nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616257(CHEMBL3605566)
Affinity DataIC50: 31nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataIC50: 39nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coliDH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616258(CHEMBL4074906)
Affinity DataIC50: 48nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 56nMAssay Description:Binding affinity to human partial length BRD4 BD1 (N44 to E168 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetThiosulfate sulfurtransferase(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50012070(CHEMBL295316 | plumbagin | 5-hydroxy-2-methylnapht...)
Affinity DataIC50: 60nMAssay Description:Inhibition of native rhodanese (unknown origin) assessed as reduction in rhodanese enzyme activity after 45 mins by Fe(SCN)3 dye based spectrometric ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616263(CHEMBL4082632)
Affinity DataIC50: 60nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 69nMAssay Description:Binding affinity to human partial length BRD3 BD1 (P24 to E144 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataIC50: 87nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coli DH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616257(CHEMBL3605566)
Affinity DataIC50: 90nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 103nMAssay Description:Binding affinity to human partial length BRD2 BD1 (K71 to N194 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 108nMAssay Description:Binding affinity to human partial length BRD3 BD2 (G306 to P416 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 119nMAssay Description:Binding affinity to human partial length BRDT BD2 (K250 to E382 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetThiosulfate sulfurtransferase(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM81348(R115 (Reactive Blue 2) | β-Lapachone (A3) | b...)
Affinity DataIC50: 120nMAssay Description:Inhibition of native rhodanese (unknown origin) assessed as reduction in rhodanese enzyme activity after 45 mins by Fe(SCN)3 dye based spectrometric ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 131nMAssay Description:Inhibition of BRD3-BD2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 142nMAssay Description:Binding affinity to human partial length BRD4 BD2 (K333 to E460 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
Target60 kDa heat shock protein, mitochondrial(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50366944(Azovan Blue | Azovan sodium | EVANS BLUE)
Affinity DataIC50: 170nMAssay Description:Inhibition of human N-terminal octa-His-tagged HSP60 expressed in Escherichia coli Rosetta(DE3) pLysS/human HSP10 expressed in Escherichia coli Roset...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616258(CHEMBL4074906)
Affinity DataIC50: 210nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50501230(CHEMBL3986320)
Affinity DataIC50: 230nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coliDH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616263(CHEMBL4082632)
Affinity DataIC50: 235nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 2(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 244nMAssay Description:Binding affinity to human partial length BRD2 BD2 (E348to D455 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetBromodomain-containing protein 3(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 262nMAssay Description:Inhibition of BRD3-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetThiosulfate sulfurtransferase(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM60918(5-Amino-2-hydroxy-benzoic acid | cid_4075 | MLS001...)
Affinity DataIC50: 280nMAssay Description:Inhibition of native rhodanese (unknown origin) assessed as reduction in rhodanese enzyme activity after 45 mins by Fe(SCN)3 dye based spectrometric ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616259(CHEMBL5412959)
Affinity DataIC50: 281nMAssay Description:Inhibition of BRD4-BD1 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50012070(CHEMBL295316 | plumbagin | 5-hydroxy-2-methylnapht...)
Affinity DataIC50: 290nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coli DH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50114392(CHEMBL3605560)
Affinity DataIC50: 294nMAssay Description:Inhibition of BRD4-BD2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetThiosulfate sulfurtransferase(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM26655(CHEMBL253570 | 2-(3,4-dihydroxyphenyl)-3,5,7,8-tet...)
Affinity DataIC50: 330nMAssay Description:Inhibition of native rhodanese (unknown origin) assessed as reduction in rhodanese enzyme activity after 45 mins by Fe(SCN)3 dye based spectrometric ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 360nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coliDH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThiosulfate sulfurtransferase(Human)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50523758(Phosphated riboflavin | Photrexa | Riboflavin 5''-...)
Affinity DataIC50: 380nMAssay Description:Inhibition of native rhodanese (unknown origin) assessed as reduction in rhodanese enzyme activity after 45 mins by Fe(SCN)3 dye based spectrometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM26655(CHEMBL253570 | 2-(3,4-dihydroxyphenyl)-3,5,7,8-tet...)
Affinity DataIC50: 390nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coli DH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBromodomain testis-specific protein(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50616255(CHEMBL3605565)
Affinity DataIC50: 403nMAssay Description:Binding affinity to human partial length BRDT BD1 (N21 to E137 residues) expressed in bacterial expression system using H4K5acIC8acK12acK16ac-biotiny...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCo-chaperonin GroES(Escherichia coli)
Indiana University School of Medicine

Curated by ChEMBL
LigandPNGBDBM23223(Tash 1 | Gossypol, 4 | 7-[8-formyl-1,6,7-trihydrox...)
Affinity DataIC50: 430nMAssay Description:Inhibition of Escherichia coli GroEL expressed in Escherichia coli DH5alpha/Escherichia coli GroES expressed in Escherichia coli BL21 (DE3) assessed ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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