Compile Data Set for Download or QSAR
Report error Found 1205 with Last Name = 'suzuki' and Initial = 'h'
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108094(CHEMBL3601200)
Affinity DataEC50:  219nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
LigandPNGBDBM50525954(CHEMBL4474443)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
LigandPNGBDBM50525957(CHEMBL4461515)
Affinity DataEC50:  49nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1B adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265530(CHEMBL4067502)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human alpha1B adrenergic receptor expressed in HEK293 cells after 6 hrs by NFAT-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  86nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.340nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 37 degC by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265528(CHEMBL4089669)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265541(CHEMBL4080868)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
LigandPNGBDBM50525942(CHEMBL4465567)
Affinity DataEC50:  663nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
LigandPNGBDBM50525952(CHEMBL4542977)
Affinity DataEC50:  670nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
LigandPNGBDBM50525945(CHEMBL4449495)
Affinity DataEC50:  125nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265532(CHEMBL4104183)
Affinity DataEC50:  6.5nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265530(CHEMBL4067502)
Affinity DataEC50:  18nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265532(CHEMBL4104183)
Affinity DataEC50:  163nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human beta2 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265529(CHEMBL4088750)
Affinity DataEC50:  309nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
LigandPNGBDBM50525956(CHEMBL4465513)
Affinity DataEC50:  1.22E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
LigandPNGBDBM50525958(CHEMBL4591600)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50095998(L-gamma-glutamyl-S-hexyl-L-cysteinylglycine | S-he...)
Affinity DataKd:  2.50E+6nMAssay Description:Binding activity towards the active site of macrophage migration inhibitory factor (MIF)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108094(CHEMBL3601200)
Affinity DataEC50:  21nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human beta1 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.490nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at recombinant human beta2 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetMacrophage migration inhibitory factor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50653054(Tp-010 | BTZO-1)
Affinity DataKd:  157nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
LigandPNGBDBM50525943(CHEMBL4449850)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
LigandPNGBDBM50525946(CHEMBL4586856)
Affinity DataEC50:  2.06E+3nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 0.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50077647(4-hydroxy-7-(1-hydroxy-2-(methylamino)ethyl)benzo[...)
Affinity DataKd:  51nMAssay Description:Compound was tested for its binding affinity to human Beta-2 adrenergic receptor by using the radioligand [3H]CGP-12177More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50525950(CHEMBL4552995)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265528(CHEMBL4089669)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human beta2 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  6nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  10nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265531(CHEMBL4105097)
Affinity DataEC50:  1.76E+3nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
LigandPNGBDBM50525953(CHEMBL4437589)
Affinity DataEC50:  60nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265529(CHEMBL4088750)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108088(CHEMBL3601305)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human alpha1A adrenergic receptor expressed in HEK293 cells assessed as intercellular Ca mobilization by Fura-2AM dye...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265542(CHEMBL4073098)
Affinity DataEC50:  18nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  23nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 4 degC by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
LigandPNGBDBM50525951(CHEMBL4447367)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108099(CHEMBL3601204)
Affinity DataEC50:  14nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at room temperature by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 0.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50156270(Methanesulfonic acid 3-(2-{2-hydroxy-2-[(R)-3-(thi...)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265530(CHEMBL4067502)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human beta1 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
TargetBeta-3 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50108091(CHEMBL3601307)
Affinity DataEC50:  66nMAssay Description:Agonist activity at recombinant human beta3 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
LigandPNGBDBM50525947(CHEMBL4560730)
Affinity DataEC50:  280nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50265528(CHEMBL4089669)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at recombinant human beta1 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 1205 total ) | Next | Last >>
Jump to: