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LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237689(CHEMBL4066943)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237692(CHEMBL4091162)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237673(CHEMBL4098085)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237682(CHEMBL4083363)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237695(CHEMBL4072935)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237701(CHEMBL4098908)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237702(CHEMBL4070220)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237698(CHEMBL4090216)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237690(CHEMBL4084928)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237688(CHEMBL4091575)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  5nMAssay Description:Inhibition of CLK1 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of CLK2 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237691(CHEMBL4080872)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237686(CHEMBL4062056)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237694(CHEMBL4061554)
Affinity DataIC50:  8nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237697(CHEMBL4085578)
Affinity DataIC50:  9.90nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237675(CHEMBL4087825)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237687(CHEMBL4083793)
Affinity DataIC50:  12nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237699(CHEMBL4060978)
Affinity DataIC50:  12nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237674(CHEMBL4099816)
Affinity DataIC50:  18nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237677(CHEMBL4062207)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237700(CHEMBL4070681)
Affinity DataIC50:  29nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237693(CHEMBL4083382)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237678(CHEMBL4082371)
Affinity DataIC50:  30nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  30nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  34nMAssay Description:Inhibition of PIM1 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  36nMAssay Description:Inhibition of CDC7 in human SW-620 cells assessed as reduction in phosphorylation of MCM2 at Ser40 residue incubated for 48 hrs by Western blot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237676(CHEMBL4066501)
Affinity DataIC50:  36nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  37nMAssay Description:Inhibition of GSK3alpha (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237696(CHEMBL4066739)
Affinity DataIC50:  44nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  51nMAssay Description:Inhibition of GSK3beta (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  53nMAssay Description:Inhibition of 1 nM AVP-induced cAMP accumulation in cells expressing human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCell division cycle 7-related protein kinase(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  53nMAssay Description:Inhibition of CDC7 in human SW-620 cells assessed as reduction in phosphorylation of MCM2 at Ser53 residue incubated for 48 hrs by Western blot analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  61nMAssay Description:Inhibition of Erk2 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  77nMAssay Description:Inhibition of PIM1 (unknown origin) pretreated for 30 mins followed by substrate addition measured after 5 hrs in presence of 1 mM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  189nMAssay Description:Inhibition of GSK3alpha (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  191nMAssay Description:ATP competitive inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  206nMAssay Description:Inhibition of CLK1 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK1(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  212nMAssay Description:Inhibition of CLK1 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  227nMAssay Description:Inhibition of CLK2 (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  251nMAssay Description:Inhibition of GSK3alpha (unknown origin) in presence of 1 mM ATP with preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK2(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50574282(CHEMBL4868568)
Affinity DataIC50:  270nMAssay Description:Inhibition of CLK2 (unknown origin) in presence of 1 mM ATP without preincubationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 3(Human)
Carna Biosciences

Curated by ChEMBL
LigandPNGBDBM50237672(CHEMBL4089159)
Affinity DataIC50:  278nMAssay Description:Inhibition of 1 nM AVP-induced calcium mobilisation in cells expressing human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237685(CHEMBL4099311)
Affinity DataIC50:  890nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237680(CHEMBL4094263)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237684(CHEMBL4081292)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237681(CHEMBL4060703)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of [3H]AVP binding to recombinant human vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237683(CHEMBL4064014)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50237679(CHEMBL4086500)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human Cdc7 (1 to 574 residues)/human N-terminal GST-tagged ASK (1 to 674 residues) expressed in baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed