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TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398475(CHEMBL2179131)
Affinity DataKi:  0.0170nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398472(CHEMBL2179138)
Affinity DataKi:  0.0360nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM16254(N2-[(2R,4S,5S)-5-{[N-{[(2,5-dimethyl-1,3-oxazol-4-...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398473(CHEMBL2179137)
Affinity DataKi:  0.400nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398471(CHEMBL2179140)
Affinity DataKi:  0.470nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398475(CHEMBL2179131)
Affinity DataIC50: 1nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM16047(EVNXXAEF | N-{(2R,4S,5S)-5-[(L-alpha-glutamyl-L-va...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of BACE1More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50231937(N-{(1S,2R)-1-benzyl-2-hydroxy-3-[(3-methoxybenzyl)...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataKi:  5.40nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398478(CHEMBL2179139)
Affinity DataKi:  7.20nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398474(CHEMBL2179136)
Affinity DataKi:  7.30nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398476(CHEMBL2179130)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 2(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398472(CHEMBL2179138)
Affinity DataKi:  11nMAssay Description:Inhibition of recombinant BACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398471(CHEMBL2179140)
Affinity DataIC50: 14nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398472(CHEMBL2179138)
Affinity DataIC50: 15nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398474(CHEMBL2179136)
Affinity DataIC50: 22nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50104413(Glutamyl-gamma-boronate analogue | CHEMBL87796)
Affinity DataKi:  25nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398480(CHEMBL2179134)
Affinity DataKi:  25nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398476(CHEMBL2179130)
Affinity DataKi:  27nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607251(CHEMBL5219012)
Affinity DataKi:  45nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607251(CHEMBL5219012)
Affinity DataKi:  77nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398477(CHEMBL2179132)
Affinity DataKi:  99nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 2(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398475(CHEMBL2179131)
Affinity DataKi:  120nMAssay Description:Inhibition of recombinant BACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398472(CHEMBL2179138)
Affinity DataKi:  530nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398473(CHEMBL2179137)
Affinity DataKi:  690nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398477(CHEMBL2179132)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of BACE1 in human neuroblastoma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398481(CHEMBL2179133)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398479(CHEMBL2179135)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of recombinant BACE1 expressed in Escherichia coli using Arg- Glu(EDANS)-Glu-Val-Asn-Leu-Asp-Ala-Glu-Phe-Lys(Dabcyl)-Arg as substrate by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetBeta-secretase 2(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398476(CHEMBL2179130)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of recombinant BACE2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398471(CHEMBL2179140)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398475(CHEMBL2179131)
Affinity DataKi:  4.30E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398474(CHEMBL2179136)
Affinity DataKi:  7.10E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetCathepsin D(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50398476(CHEMBL2179130)
Affinity DataKi:  8.26E+3nMAssay Description:Inhibition of human cathepsin DMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607252(CHEMBL5219273)
Affinity DataKi:  2.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607253(CHEMBL5220603)
Affinity DataKi:  4.60E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607257(CHEMBL5219724)
Affinity DataKi:  4.90E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607262(CHEMBL5218792)
Affinity DataKi:  6.10E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607252(CHEMBL5219273)
Affinity DataKi:  8.70E+4nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607258(CHEMBL5218962)
Affinity DataKi:  8.80E+4nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607257(CHEMBL5219724)
Affinity DataKi:  1.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607261(CHEMBL5218489)
Affinity DataKi:  1.73E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607255(CHEMBL5219778)
Affinity DataKi:  2.02E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607256(CHEMBL5220724)
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607254(CHEMBL5219218)
Affinity DataKi:  2.54E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607253(CHEMBL5220603)
Affinity DataKi:  2.60E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607259(CHEMBL5220006)
Affinity DataKi:  3.43E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607256(CHEMBL5220724)
Affinity DataKi:  3.56E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607258(CHEMBL5218962)
Affinity DataKi:  5.08E+5nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607260(CHEMBL5218520)
Affinity DataKi:  5.89E+5nMAssay Description:Inhibition of human GGT1 transpeptidation in Pichia pastoris using L-GpNA as substrate in presence of Gly-GlyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlutathione hydrolase 1 proenzyme(Human)
State University of New York

Curated by ChEMBL
LigandPNGBDBM50607254(CHEMBL5219218)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human GGT1 expressed in Pichia pastoris assessed as inhibition of GSH hydrolysis measured by L-glutamate release assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
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