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TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50074569(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  1.00E+3nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473895(CHEMBL285811)
Affinity DataEC50:  324nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473896(CHEMBL126103)
Affinity DataEC50:  170nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473897(CHEMBL126655)
Affinity DataEC50:  135nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473898(CHEMBL126199)
Affinity DataEC50:  178nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473899(CHEMBL262632)
Affinity DataEC50:  47nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473900(CHEMBL124330)
Affinity DataEC50:  36nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473901(CHEMBL122499)
Affinity DataEC50:  55nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50473902(CHEMBL127933)
Affinity DataEC50:  71nMAssay Description:Binding of [3H]N-methylscopolamine at porcine heart Muscarinic acetylcholine receptor M2 that inhibits the dissociation of [3H]NMS half maximally (pE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474518(CHEMBL9017)
Affinity DataEC50:  447nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474519(CHEMBL8900)
Affinity DataEC50:  309nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473896(CHEMBL126103)
Affinity DataEC50:  170nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474520(CHEMBL216974)
Affinity DataEC50:  204nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474521(CHEMBL8763)
Affinity DataEC50:  6.31E+3nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474522(CHEMBL8669)
Affinity DataEC50:  457nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474523(CHEMBL8532)
Affinity DataEC50:  8.5nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474524(CHEMBL406431)
Affinity DataEC50:  36nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474525(CHEMBL418702)
Affinity DataEC50:  398nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473900(CHEMBL124330)
Affinity DataEC50:  36nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474526(CHEMBL269592)
Affinity DataEC50:  7.80nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473898(CHEMBL126199)
Affinity DataEC50:  178nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474527(CHEMBL262448)
Affinity DataEC50:  115nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473897(CHEMBL126655)
Affinity DataEC50:  135nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473902(CHEMBL127933)
Affinity DataEC50:  71nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474528(CHEMBL8764)
Affinity DataEC50:  204nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474529(CHEMBL8449)
Affinity DataEC50:  25nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474530(CHEMBL269205)
Affinity DataEC50:  145nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474531(CHEMBL7902)
Affinity DataEC50:  501nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474532(CHEMBL275988)
Affinity DataEC50:  1.62E+3nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM80806(3-[1,3-bis(oxidanylidene)benzo[de]isoquinolin-2-yl...)
Affinity DataEC50:  14nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50074569(Bis-{3-(1,3-dioxo-2,3-dihydro-1H-2-isoindolyl)prop...)
Affinity DataEC50:  1.35E+3nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474533(CHEMBL268195)
Affinity DataEC50:  741nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473895(CHEMBL285811)
Affinity DataEC50:  324nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474534(CHEMBL8518)
Affinity DataEC50:  52nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474535(CHEMBL8721)
Affinity DataEC50:  14nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474536(CHEMBL274564)
Affinity DataEC50:  19nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474537(CHEMBL262449)
Affinity DataEC50:  302nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473899(CHEMBL262632)
Affinity DataEC50:  47nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50473901(CHEMBL122499)
Affinity DataEC50:  55nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474538(CHEMBL406691)
Affinity DataEC50:  7.60nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50448376(Naphmethonium)
Affinity DataEC50:  4.40nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474539(CHEMBL273255)
Affinity DataEC50:  120nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474540(CHEMBL8855)
Affinity DataEC50:  229nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Pig)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50474541(CHEMBL8653)
Affinity DataEC50:  115nMAssay Description:Effective concentration required to inhibit dissociation of [3H]NMS from porcine heart ventricles muscarinic acetylcholine receptor M2.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50220060((14-dimethylaminomethyl-6H,13H-pyrazino[1,2-a;4,5-...)
Affinity DataEC50:  1.66E+4nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in hepes bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50220060((14-dimethylaminomethyl-6H,13H-pyrazino[1,2-a;4,5-...)
Affinity DataEC50:  447nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in Na,K,Pi bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50475689(4,4''-Dimethylcaracurinium V Dichloride | Dimethyl...)
Affinity DataEC50:  8.10nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in Na,K,Pi bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50025037(CHEBI:3382 | Caracurine V)
Affinity DataEC50:  437nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in Na,K,Pi bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50220046(trimethyl({20-[(trimethylazaniumyl)methyl]-3,13-di...)
Affinity DataEC50:  1.12E+4nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in hepes bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Human)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50220045([(20-{[dimethyl(prop-2-en-1-yl)azaniumyl]methyl}-3...)
Affinity DataEC50:  110nMAssay Description:Inhibition of [3H]NMS dissociation from muscarinic M2 receptor in Na,K,Pi bufferMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
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