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TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463552(CHEMBL4249862)
Affinity DataEC50:  2.20E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50386790(CHEMBL1829174 | CHEMBL2047159 | TAK-875 | US119052...)
Affinity DataEC50:  5.10E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463553(CHEMBL4248812)
Affinity DataEC50:  4.00E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463554(CHEMBL4244619)
Affinity DataEC50:  800nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463555(CHEMBL4241897)
Affinity DataEC50:  800nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463556(CHEMBL4238097)
Affinity DataEC50:  5.40E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463557(CHEMBL4248694)
Affinity DataEC50:  1.20E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50463558(CHEMBL4241974)
Affinity DataEC50:  3.00E+3nMAssay Description:Transactivation of human GPR40 expressed in HEK293 cells after 24 hrs by Elk-Gal4 luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550968(CHEMBL4743350)
Affinity DataEC50:  3.13E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550969(CHEMBL4744389)
Affinity DataEC50:  600nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550970(CHEMBL4750433)
Affinity DataEC50:  830nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550973(CHEMBL4784857)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550974(CHEMBL4795875)
Affinity DataEC50:  1.93E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550977(CHEMBL4740282)
Affinity DataEC50:  650nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550978(CHEMBL4782382)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50244791((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)
Affinity DataEC50:  640nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550979(CHEMBL4785060)
Affinity DataEC50:  2.56E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550980(CHEMBL4745258)
Affinity DataEC50:  3.99E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550981(CHEMBL4776485)
Affinity DataEC50:  1.85E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550982(CHEMBL4764779)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550983(CHEMBL4749117)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Chinese Academy of Medical Sciences&Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50550984(CHEMBL4751384)
Affinity DataEC50:  4.02E+3nMAssay Description:Agonist activity at CREB-LBD and Gal4-DBD fused recombinant human GPR119 expressed in HEK293 cells by firefly luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50551529(CHEMBL4785863)
Affinity DataKd:  4.80E+3nMAssay Description:Binding affinity to immobilized human 20S proteasome beta 5 subunit by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetProteasome subunit beta type-5(Human)
Peking University Health Science Center

Curated by ChEMBL
LigandPNGBDBM50551532(CHEMBL4744709)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to immobilized human 20S proteasome beta 5 subunit by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2022
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425793(CHEMBL2316881)
Affinity DataKd:  2.95E+3nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425794(CHEMBL2316883)
Affinity DataKd:  222nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425795(CHEMBL2316882)
Affinity DataKd:  1.20E+4nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425796(CHEMBL2316884)
Affinity DataKd:  175nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425797(CHEMBL2316885)
Affinity DataKd:  19nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425798(CHEMBL2316886)
Affinity DataKd:  68nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425799(CHEMBL2316888)
Affinity DataKd:  850nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425800(CHEMBL2316887)
Affinity DataKd:  3.60E+5nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425801(CHEMBL2316891)
Affinity DataKd:  1.37E+5nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425805(CHEMBL2316890)
Affinity DataKd:  1.90E+6nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425803(CHEMBL2316893)
Affinity DataKd:  1.30E+6nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50425804(6-Phenylnicotinic Acid | CHEMBL2316892)
Affinity DataKd:  2.30E+6nMAssay Description:Binding affinity to human LDH-A by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145918(CHEMBL3763993)
Affinity DataKd:  1.32E+5nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145919(CHEMBL3765610)
Affinity DataKd:  1.94E+5nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145918(CHEMBL3763993)
Affinity DataKd:  4.90E+5nMAssay Description:Binding affinity to carbonic anhydrase2 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145921(CHEMBL3763196)
Affinity DataKd:  3.40E+5nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145921(CHEMBL3763196)
Affinity DataKd:  1.40E+6nMAssay Description:Binding affinity to carbonic anhydrase2 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145925(CHEMBL3764475)
Affinity DataKd:  6.30E+5nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145925(CHEMBL3764475)
Affinity DataKd:  6.70E+5nMAssay Description:Binding affinity to carbonic anhydrase2 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145927(CHEMBL3764395)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145928(CHEMBL3765077)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145929(CHEMBL3765650)
Affinity DataKd:  4.30E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145930(CHEMBL3763340)
Affinity DataKd:  3.70E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145931(CHEMBL3764898)
Affinity DataKd:  769nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145934(CHEMBL3764904)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
TargetCholine kinase alpha(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50145939(CHEMBL3764767)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to human N-terminal truncated ChoKalpha1 (75 to 457 residues) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/15/2017
Entry Details Article
PubMed
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