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TargetMitogen-activated protein kinase 7(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  160nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  120nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  420nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  1.00E+3nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  480nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Harvard Medical School

LigandPNGBDBM81377(FIIN-1)
Affinity DataKd:  210nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase Blk(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  2.30E+3nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 7(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  130nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  3.10nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 2(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  5.60nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 3(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  5.40nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 4(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  280nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  49nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  340nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  250nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  1.40E+3nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  480nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Harvard Medical School

LigandPNGBDBM81378(FRIN-1)
Affinity DataKd:  470nMAssay Description:In vitro kinase assay profiled against a panel of different kinase binding assay using Ambit kinomeScan technology. Biochemical IC50 values were det...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ABL1(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  3.30nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  1.20nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase B-raf(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  36nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetCyclin-dependent kinase 11B(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  32nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetCyclin-dependent kinase 2(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  840nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetCyclin-dependent kinase 3(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  250nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetCyclin-dependent kinase 5(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  150nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetCyclin-dependent kinase 7(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  13nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  3.40nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 1(Human)
Harvard Medical School

LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  74nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  2.30nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 3(Human)
Harvard Medical School

LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  31nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetHomeodomain-interacting protein kinase 1(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  34nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetMast/stem cell growth factor receptor Kit(Human)
Harvard Medical School

LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  2.90nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetSerine/threonine-protein kinase 10(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  9.5nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 12(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  100nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetPlatelet-derived growth factor receptor alpha(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  7.70nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetPlatelet-derived growth factor receptor beta(Rat)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  1.80nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  5.60nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetAngiopoietin-1 receptor(Human)
Dana-Farber Cancer Institute

US Patent
LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  57nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetVascular endothelial growth factor receptor 2(Human)
Harvard Medical School

LigandPNGBDBM124970(US8765747, 2)
Affinity DataKd:  58nMAssay Description:KINOMEscan (Ambit Biosciences, San Diego, Calif.), a high-throughput method for screening small molecular agents against a large panel of human kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/18/2014
Entry Details
Go to US Patent

TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271300(CHEMBL4125758 | US12012467, Compound DI-39)
Affinity DataKd:  56nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271349(CHEMBL4128744 | US12012467, Compound DI-68)
Affinity DataKd:  32nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271350(CHEMBL4128331 | US12012467, Compound DI-67)
Affinity DataKd:  37nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271312(CHEMBL4129556 | US12012467, Compound DI-64)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271359(CHEMBL4128753 | US12012467, Compound DI-71)
Affinity DataKd:  8.30nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271360(CHEMBL4128590 | US12012467, Compound DI-70)
Affinity DataKd:  4.10nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271361(CHEMBL4127438 | US12012467, Compound DI-404)
Affinity DataKd:  6.70nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271362(CHEMBL4126395 | US12012467, Compound DI-417)
Affinity DataKd:  1.47E+3nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetDCN1-like protein 1(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50271364(CHEMBL4129669 | US12012467, Compound DI-431)
Affinity DataKd:  5.70nMAssay Description:Binding affinity to biotin labeled recombinant N-terminal His6-tagged human DCN1 (58 to 259 residues) expressed in Escherichia coli Rosetta2 cells by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Merck Research Laboratory

Curated by ChEMBL
LigandPNGBDBM50458655(CHEMBL4207377)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human CRTh2 expressed in HEK cells assessed as forskolin-induced intracellular cAMP accumulation by ELISA based chemiluminescence...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha/Vitamin D3 receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50469127(CHEMBL4288947)
Affinity DataEC50:  6.40nMAssay Description:Transactivation of recombinant human VDR/RXRalpha expressed in HEK293 cells after 24 hrs by Dual-luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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