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TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  316nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50:  794nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50: <2.00E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50:  5.01E+4nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497461(CHEMBL3343990)
Affinity DataEC50:  501nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497462(CHEMBL3343987)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50:  501nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50:  3.16E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  316nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497458(CHEMBL3343994)
Affinity DataEC50:  631nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497460(CHEMBL3343988)
Affinity DataEC50:  3.98E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50412987(CHEMBL475965)
Affinity DataEC50: <2.00E+3nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497464(CHEMBL3343993)
Affinity DataEC50:  1.58E+4nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Mouse)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM224021(BAM8-22 | VGRPEWWMDYQKRYG)
Affinity DataEC50:  251nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497463(CHEMBL3343991)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50497459(CHEMBL3343992)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Rat)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50336912(Adamantane-1-carboxylic acid [(S)-1-((S)-1-carbamo...)
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075195(CHEMBL3414847)
Affinity DataKd:  166nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50313638(1-(4-methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-c...)
Affinity DataKd:  5.50E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataEC50:  372nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50448377(CHEMBL3121473)
Affinity DataEC50:  2nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50008072((3S-cis)-3-ethyldihydro-4-[(1-methyl-1H-imidazol-5...)
Affinity DataEC50:  832nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075196(CHEMBL3414838)
Affinity DataEC50:  58nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075197(CHEMBL3414839)
Affinity DataEC50:  63nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075198(CHEMBL3414840)
Affinity DataEC50:  32nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075199(CHEMBL3414841)
Affinity DataEC50:  178nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075200(CHEMBL3414842)
Affinity DataEC50:  15nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075201(CHEMBL3414843)
Affinity DataEC50:  302nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075202(CHEMBL3414844)
Affinity DataEC50:  59nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075203(CHEMBL3414845)
Affinity DataEC50:  537nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50075195(CHEMBL3414847)
Affinity DataEC50:  60nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50313638(1-(4-methoxybenzyl)-4-oxo-1,4-dihydroquinoline-3-c...)
Affinity DataEC50:  8.32E+3nMAssay Description:Partial agonist activity at human muscarinic M1 acetylcholine receptor expressed in CHO cells assessed as increase in IP1 accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM10759(2-acetoxyethyl(trimethyl)ammonium;perchlorate | 2-...)
Affinity DataKd:  1.74E+4nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50448377(CHEMBL3121473)
Affinity DataKd:  2.14E+3nMAssay Description:Displacement of [3H]NMS from human muscarinic M1 acetylcholine receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
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