Affinity DataIC50: 1.80nMAssay Description:Binding affinity towards Cannabinoid receptor 1 was determined using [3H]-CP- cannabinoid as radioligand with mouse brain memebraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.90nMAssay Description:Agonist activity at CB1 receptor in field-stimulated mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of radioligand from CB1 receptor in mouse brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]CP55940 from mouse CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 6.90nMAssay Description:Binding affinity towards Cannabinoid receptor 1 was determined using [3H]-CP- cannabinoid as radioligand with mouse brain memebraneMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brainMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Partial agonist activity at mouse CB1 receptor by vas deferens assayMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Binding affinity towards Cannabinoid receptor 1 was determined using [3H]-CP- cannabinoid as radioligand with mouse brain memebrane in the presence o...More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Allosteric antagonist activity at mouse CB1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Allosteric antagonist activity at mouse CB1 receptor by GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Agonist activity at CB1 receptor in mouse Neuro2a cells assessed as inhibition of forskolin-stimulated adenylyl cyclase activity after 15 mins by liq...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:A functional assay screen for the inhibition of adenylate cyclase (AC) activity was chosen as the subsequent assay. This screen would allow us to gai...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 1 uM CP55,940-induced [35S]GTPgammaS binding i...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 1 uM CP55,940-induced [35S]GTPgammaS binding i...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 1 uM CP55,940-induced [35S]GTPgammaS binding i...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 1 uM CP55,940-induced [35S]GTPgammaS binding i...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 100 nM CP55,940-induced [35S]GTPgammaS binding...More data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Allosteric modulator activity at CB1 receptor in mouse cerebellar membranes assessed as suppression of 100 nM CP55,940-induced [35S]GTPgammaS binding...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 76nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: 97nMAssay Description:Inverse agonist at mouse brain CB1R expressed in CHOK1 cell membranes assessed as inhibition of CP55940-stimulated [35S]GTP-gammaS binding measured a...More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: <100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair