Compile Data Set for Download or QSAR
maximum 50k data
Found 11 of kd data for polymerid = 1277
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12016(2,3-difluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,3-DIFLU...)
Affinity DataKd:  1.60nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12023(2,3,4,5,6-pentafluoro-SBB | 4-(AMINOSULFONYL)-N-[(...)
Affinity DataKd:  2nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12018(2,5-difluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,5-DIFLU...)
Affinity DataKd:  2.20nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12014(2-fluoro-SBB | 4-(AMINOSULFONYL)-N-[(2-FLUOROPHENY...)
Affinity DataKd:  2.30nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12017(2,4-difluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,4-DIFLU...)
Affinity DataKd:  3.30nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12015(4-(AMINOSULFONYL)-N-[(4-FLUOROPHENYL)METHYL]-BENZA...)
Affinity DataKd:  3.30nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12020(2,3,4-trifluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,3,4-...)
Affinity DataKd:  3.80nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12019(2,6-difluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,6-DIFLU...)
Affinity DataKd:  3.90nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12021(2,4,6-trifluoro-SBB | 4-(AMINOSULFONYL)-N-[(2,4,6-...)
Affinity DataKd:  3.90nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12022(3,4,5-trifluoro-SBB | 4-(AMINOSULFONYL)-N-[(3,4,5-...)
Affinity DataKd:  3.90nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair
TargetCarbonic anhydrase 2 [F130V](Homo sapiens (Human))
University Of Pennsylvania

LigandPNGBDBM12013(4-(AMINOSULFONYL)-N-PHENYLMETHYLBENZAMIDE | CHEMBL...)
Affinity DataKd:  5.60nMpH: 7.4 T: 2°CAssay Description:Inhibitor binding to CA II was determined using a fluorescence competition assay. Displacement of dansylamide and binding of the inhibitor was determ...More data for this Ligand-Target Pair