Compile Data Set for Download or QSAR
Report error Found 59 of ic50 data for polymerid = 2131
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018697BDBM50018697(CHEMBL3291310)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095604BDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018695BDBM50018695(CHEMBL3291308)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 571388BDBM571388(US11440916, HZ10136)
Affinity DataIC50: 1.10nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202993BDBM50202993(2-furan-2-yl-7-[2-(4-phenyl-piperazin-1-yl)-ethyl]...)
Affinity DataIC50: 1.20nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039676BDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50048466BDBM50048466(CHEMBL17127 | SCH58261 | 2-(furan-2-yl)-7-phenethy...)
Affinity DataIC50: 1.80nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018693BDBM50018693(CHEMBL3291306)
Affinity DataIC50: 1.90nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50202986BDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataIC50: 2.5nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095602BDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018696BDBM50018696(CHEMBL3291309)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004566BDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018692BDBM50018692(CHEMBL3291305)
Affinity DataIC50: 3.60nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053927BDBM50053927(7-Methyl-2-phenyl-4-((E)-styryl)-1,4-dihydro-quino...)
Affinity DataIC50: 4.77nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018688BDBM50018688(CHEMBL3291301)
Affinity DataIC50: 5.10nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018689BDBM50018689(CHEMBL3291302)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 7.05nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50382493BDBM50382493(CHEMBL2024116)
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 0.1 uM adenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095605BDBM50095605(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095606BDBM50095606(4-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetrahy...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50095603BDBM50095603(4-[5-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataIC50: 10nMAssay Description:Inhibition of [3H]ZM-241385 binding to adenosine A2A receptor(AR).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275963BDBM50275963((S)-N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(3-fluor...)
Affinity DataIC50: 15nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018691BDBM50018691(CHEMBL3291304)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009546BDBM50009546(CHEMBL98637 | 2-{6-Amino-2-[2-(4-methoxy-phenyl)-e...)
Affinity DataIC50: 23nMAssay Description:Binding affinity for Adenosine A2A receptor using [3H]ZM-24138 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 26236BDBM26236(CHEMBL487569 | N-[6-(3,5-dimethoxyphenyl)-2-(3,5-d...)
Affinity DataIC50: 29nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275803BDBM50275803(N-(2-(3,5-dimethyl-1H-pyrazol-1-yl)-6-(3-(1-methyl...)
Affinity DataIC50: 42nMAssay Description:Activity at adenosine A2A receptor in rat PC12 cells assessed as intracellular cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 86760BDBM86760(CAS_104924 | NSC_104924 | CGS 21680 | US11440916, ...)
Affinity DataIC50: 66.9nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50009531BDBM50009531(CHEMBL2112337 | 2-[6-Amino-2-(2-phenyl-propylamino...)
Affinity DataIC50: 68nMAssay Description:Binding affinity against Adenosine A2A receptor in rat striatal membranes b displacement of [3H]-CGS- 21680More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018690BDBM50018690(CHEMBL3291303)
Affinity DataIC50: 76nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018694BDBM50018694(CHEMBL3291307)
Affinity DataIC50: 97nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50382493BDBM50382493(CHEMBL2024116)
Affinity DataIC50: 97nMAssay Description:Antagonist activity at rat adenosine 2A receptor assessed as reduction in cAMP level in presence of 10 uM adenosineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50450928BDBM50450928(CHEMBL2113728)
Affinity DataIC50: 100nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50053924BDBM50053924(CHEMBL89093 | MRS1067 | 3,6-Dichloro-2-(2-isopropo...)
Affinity DataIC50: 100nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018683BDBM50018683(CHEMBL3291296)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50176050BDBM50176050(8-(3,4-dimethoxystyryl)-1,3-diethyl-7-methyl-1H-pu...)
Affinity DataIC50: 228nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393188BDBM50393188(CHEMBL2153620)
Affinity DataIC50: 251nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptor in presence of 100 mM NaClMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50393188BDBM50393188(CHEMBL2153620)
Affinity DataIC50: 263nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21220BDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataIC50: 366nMAssay Description:Displacement of [3H]MSX-2 from rat adenosine A2A receptor in presence of 100 mM NaClMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50023498BDBM50023498(2-(5-Bromo-furan-2-yl)-9-chloro-[1,2,4]triazolo[1,...)
Affinity DataIC50: 531nMAssay Description:Binding affinity for Adenosine A2A receptor from rat striatal membranes using [3H]-CGH 21680More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50531422BDBM50531422(CHEMBL4522981)
Affinity DataIC50: 750nMAssay Description:Antagonist activity at recombinant rat A2A adenosine receptor expressed in CHO cells after 3 to 4 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079655BDBM50079655({2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)...)
Affinity DataIC50: 840nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21173BDBM21173(DPCPX | CHEMBL183 | 8-cyclopentyl-1,3-dipropyl-2,3...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50208945BDBM50208945(N6-(4-hydroxybenzyl)adenine riboside | CHEMBL22402...)
Affinity DataIC50: 4.66E+3nMAssay Description:Binding affinity to adenosine A2A receptor in rat brain striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50450927BDBM50450927(CHEMBL2113729)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079649BDBM50079649({2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079654BDBM50079654(4-(6-oxo-3-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)py...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50079650BDBM50079650({2-[6-Oxo-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibitory activity against Adenosine A2a receptor using [3H]NECA in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018680BDBM50018680(CHEMBL3291293)
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018679BDBM50018679(CHEMBL3291292)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
Yamasa

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50018682BDBM50018682(CHEMBL3291295)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at adenosine A2A receptor in 5-HT-treated Wistar rat femoral vein assessed as inhibition of 2-octyn-1-yladenosine-induced vasodil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/11/2015
Entry Details Article
PubMed
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