Compile Data Set for Download or QSAR
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TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622583(CHEMBL5413450)
Affinity DataEC50:  0.0500nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622574(CHEMBL5413099)
Affinity DataEC50: <0.100nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622567(CHEMBL5406029)
Affinity DataEC50:  0.200nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622570(CHEMBL5409708)
Affinity DataEC50:  0.200nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622569(CHEMBL5426454)
Affinity DataEC50:  0.200nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622572(CHEMBL5437022)
Affinity DataEC50:  0.200nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622576(CHEMBL5405858)
Affinity DataEC50:  0.200nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622581(CHEMBL5402691)
Affinity DataEC50:  0.300nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622565(CHEMBL5439670)
Affinity DataEC50:  0.600nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622571(CHEMBL5395475)
Affinity DataEC50:  0.600nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622582(CHEMBL5397398)
Affinity DataEC50:  1nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622564(CHEMBL5438596)
Affinity DataEC50:  1nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622573(CHEMBL5419387)
Affinity DataEC50:  1.10nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622562(CHEMBL5412027)
Affinity DataEC50:  1.20nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622563(CHEMBL5405240)
Affinity DataEC50:  1.30nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622579(CHEMBL5429111)
Affinity DataEC50:  1.70nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622561(CHEMBL5397498)
Affinity DataEC50:  1.70nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622575(CHEMBL5433043)
Affinity DataEC50:  1.80nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607602(CHEMBL5220994)
Affinity DataEC50:  3.20nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622568(CHEMBL5418675)
Affinity DataEC50:  3.30nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622577(CHEMBL5419069)
Affinity DataEC50:  3.70nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622580(CHEMBL5405265)
Affinity DataEC50:  4.80nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607601(CHEMBL5219667)
Affinity DataEC50:  6.30nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453957(CHEMBL4217213)
Affinity DataEC50:  6.60nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50269847(CHEMBL4097025)
Affinity DataEC50:  6.60nMAssay Description:Inhibition of CBP in human MV-4-11 cells assessed as decrease in MYC expression incubated for 4 hrs measured by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607605(CHEMBL5219177)
Affinity DataEC50:  7.90nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622566(CHEMBL5434991)
Affinity DataEC50:  12nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50250911(CHEMBL4095153 | US10696655, Example 45 | US1116807...)
Affinity DataEC50:  12nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as reduction in MYC expression after 4 hrs by luminescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2019
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607593(CHEMBL5219693)
Affinity DataEC50:  13nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50269849(CHEMBL4076748)
Affinity DataEC50:  14nMAssay Description:Inhibition of CBP in human MV-4-11 cells assessed as decrease in MYC expression incubated for 4 hrs measured by luminescence methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607600(CHEMBL5220956)
Affinity DataEC50:  16nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453949(CHEMBL4208820 | US11247989, Example 87)
Affinity DataEC50:  18nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453950(CHEMBL4203082 | US11247989, Example 88)
Affinity DataEC50:  32nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607596(CHEMBL5221053)
Affinity DataEC50:  40nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50622578(CHEMBL5431340)
Affinity DataEC50:  40nMAssay Description:Induction of CBP degradation in human RS4-11 cells incubated for 4 hrs by Western blot assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607595(CHEMBL5219030)
Affinity DataEC50:  50nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607599(CHEMBL5220732)
Affinity DataEC50:  50nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50250892(CHEMBL4061254 | US10696655, Example 63 | US1116807...)
Affinity DataEC50:  53nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as reduction in MYC expression after 4 hrs by luminescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2019
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataEC50:  69nMAssay Description:Inhibition of CBP/EP300 in human MOLM16 cells assessed as decrease in MYC expression measured after 4 hrs by RT-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453948(CHEMBL4204490 | US11247989, Example 96)
Affinity DataEC50:  76nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607598(CHEMBL5220447)
Affinity DataEC50:  79nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607597(CHEMBL5219157)
Affinity DataEC50:  100nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453970(CHEMBL4207965 | US11247989, Example 98)
Affinity DataEC50:  110nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607590(CHEMBL5220332)
Affinity DataEC50:  200nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453976(CHEMBL4209361 | US11247989, Example 97)
Affinity DataEC50:  220nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607585(CHEMBL5219512)
Affinity DataEC50:  251nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50453971(CHEMBL4204065 | US11247989, Example 11)
Affinity DataEC50:  280nMAssay Description:Inhibition of P300/CBP in human MV4-11 cells assessed as downregulation of MYC expressionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50178219(CHEMBL3814752)
Affinity DataEC50:  300nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to CBP (unknown origin) expressed in HEK293 cells after overnight incubation by luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/17/2017
Entry Details Article
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607586(CHEMBL5221030)
Affinity DataEC50:  316nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCREB-binding protein/Histone acetyltransferase p300(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50607589(CHEMBL5219678)
Affinity DataEC50:  316nMAssay Description:Inhibition of CBP/p300 in human COLO 320HSR cells assessed as reduction of C-myc levels measured after 24 hrs by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
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