Compile Data Set for Download or QSAR
Report error Found 8 of ki data for polymerid = 436
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407493BDBM50407493(CHEMBL5288446)
Affinity DataKi:  15nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50369190BDBM50369190(CHEMBL4163133)
Affinity DataKi:  15nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407492BDBM50407492(CHEMBL5280732)
Affinity DataKi:  120nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407464BDBM50407464(CHEMBL5289275)
Affinity DataKi:  2.41E+3nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407467BDBM50407467(CHEMBL5289169)
Affinity DataKi:  3.12E+3nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407491BDBM50407491(CHEMBL5282293)
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50481595BDBM50481595(CHEMBL5287183)
Affinity DataKi:  4.46E+4nMAssay Description:Binding affinity to APC (unknown origin) assessed as inhibition constant by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAdenomatous polyposis coli protein(Human)
Gitam (Deemed To Be University)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50407461BDBM50407461(CHEMBL5274458)
Affinity DataKi:  4.46E+4nMAssay Description:Inhibition of APC (303 to 739 residues) (unknown origin) assessed as inhibition constant preincubated for 60 mins followed by substrate addition and ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed