Compile Data Set for Download or QSAR
Report error Found 35 of kd for UniProtKB: Q96P20
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataKd:  0.532nMAssay Description:Binding affinity to NLRP3 (unknown origin) expressed in HEK293T cells incubated for 30 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622947BDBM50622947(CHEMBL5430191 | US20250243172, Compound Formula IX...)
Affinity DataKd:  0.860nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622943BDBM50622943(CHEMBL5409713 | US20250243172, Compound Formula V ...)
Affinity DataKd:  0.980nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622944BDBM50622944(CHEMBL5402231 | US20250243172, Compound Formula VI...)
Affinity DataKd:  3nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565841BDBM50565841(CHEMBL4795253)
Affinity DataKd:  8.80nMAssay Description:Binding affinity to biotinylated human recombinant NLRP3 PYD domain by biolayer interferometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50636762BDBM50636762(CHEMBL5567870)
Affinity DataKd:  11nMAssay Description:Binding affinity to NLRP3 (unknown origin) expressed in HEK293T cells incubated for 30 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataKd:  18nMAssay Description:Binding affinity to human NLRP3 by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647995BDBM50647995(CHEMBL5597392)
Affinity DataKd:  18nMAssay Description:Binding affinity to human NLRP3 by SPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622941BDBM50622941(CHEMBL5417338)
Affinity DataKd:  18nMAssay Description:Binding affinity to full-length human recombinant NLRP3 assessed as dissociation constant incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50634191BDBM50634191(CHEMBL5397385)
Affinity DataKd:  21nMAssay Description:Binding affinity to GFP-flag-tagged human NLRP3 transfected in HEK293T cells assessed as equilibrium dissociation constant measured after 40 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622942BDBM50622942(CHEMBL5400432)
Affinity DataKd:  24nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622941BDBM50622941(CHEMBL5417338)
Affinity DataKd:  25nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataKd:  38nMAssay Description:Binding affinity to human recombinant NLRP3 (1 to 1036 residues) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622948BDBM50622948(CHEMBL5434916 | US20250243172, Compound Formula X ...)
Affinity DataKd:  55nMAssay Description:Binding affinity to full-length human recombinant NLRP3 assessed as dissociation constant incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622948BDBM50622948(CHEMBL5434916 | US20250243172, Compound Formula X ...)
Affinity DataKd:  69nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50598211BDBM50598211(CHEMBL5173327)
Affinity DataKd:  84nMAssay Description:Binding affinity to human recombinant full length NLRP3 transfected in HEK293F cells assessed as dissociation constant incubated for 40 mins by micro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50631252BDBM50631252(CHEMBL5413950)
Affinity DataKd:  103nMAssay Description:Binding affinity to human NLRP3 assessed as equilibrium dissociation constant by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646291BDBM50646291(CHEMBL5594893)
Affinity DataKd:  104nMAssay Description:Binding affinity to streptavidin sensor chip-immobilized biotinylated recombinant human NLRP3 NACHT domain extracted from Sf9 insect cells assessed a...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50629371BDBM50629371(CHEMBL5439097)
Affinity DataKd:  110nMAssay Description:Binding affinity to human recombinant NLRP3 (1 to 1036 residues) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50605172BDBM50605172(CHEMBL5202921)
Affinity DataKd:  213nMAssay Description:Binding affinity to GFP-fused NLRP3 (unknown origin) expressed in HEK293T cells by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/25/2023
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575103BDBM50575103(CHEMBL4849582)
Affinity DataKd:  263nMAssay Description:Binding affinity to His-GFP fused tagged NLRP3 (unknown origin) expressed in HEK293T incubated for 30 mins by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622946BDBM50622946(CHEMBL5423405 | US20250243172, Compound Formula VI...)
Affinity DataKd:  480nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50622945BDBM50622945(CHEMBL5435765)
Affinity DataKd:  700nMAssay Description:Binding affinity to human recombinant NLRP3 inflammasomeMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50646422BDBM50646422(CHEMBL5584083)
Affinity DataKd:  929nMAssay Description:Binding affinity to CM5 chip-immobilized NLRP3 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647121BDBM50647121(CHEMBL5591066)
Affinity DataKd:  1.05E+3nMAssay Description:Binding affinity to human NLRP3 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635585BDBM50635585(CHEMBL5555568)
Affinity DataKd:  1.61E+3nMAssay Description:Binding affinity to LRR domain of NLRP3 (unknown origin) assessed as equilibrium dissociation constant by biolayer interferometry (BLI) analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50638473BDBM50638473(CHEMBL5556215)
Affinity DataKd:  4.34E+3nMAssay Description:Binding affinity to biotinylated NLRP3 NACHT domain (unknown origin) assessed as dissociation constant by Biolayer Interferometry assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635591BDBM50635591(CHEMBL5542846)
Affinity DataKd:  6.11E+3nMAssay Description:Binding affinity to LRR domain of NLRP3 (unknown origin) by isothermal titration calorimetry (ITC) analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635585BDBM50635585(CHEMBL5555568)
Affinity DataKd:  6.41E+3nMAssay Description:Binding affinity to LRR domain of NLRP3 (unknown origin) by isothermal titration calorimetry (ITC) analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50638473BDBM50638473(CHEMBL5556215)
Affinity DataKd:  6.82E+3nMAssay Description:Binding affinity to biotinylated NLRP3 PYD domain (unknown origin) assessed as dissociation constant by Biolayer Interferometry assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50652000BDBM50652000(CHEMBL5639831)
Affinity DataKd:  7.20E+3nMAssay Description:Binding affinity to CM5 chip immobilized NLRP3 (unknown origin) assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565841BDBM50565841(CHEMBL4795253)
Affinity DataKd:  1.72E+4nMAssay Description:Binding affinity to biotinylated human recombinant NLRP3 NACHT domain by biolayer interferometry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635579BDBM50635579(CHEMBL5555880)
Affinity DataKd:  1.85E+4nMAssay Description:Binding affinity to human LRR domain of NLRP3 assessed as dissociation constant by isothermal titration calorimetry (ITC) methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50635585BDBM50635585(CHEMBL5555568)
Affinity DataKd:  8.81E+4nMAssay Description:Binding affinity to NACHT domain of NLRP3 (unknown origin) assessed as equilibrium dissociation constant by biolayer interferometry (BLI) analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50597920BDBM50597920(CHEMBL5180041)
Affinity DataKd:  1.63E+6nMAssay Description:Binding affinity to recombinant human full length NLRP3 expressed in Sf9 insect cells assessed as dissociation constant incubated for 30 mins by MST ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed