Compile Data Set for Download or QSAR
maximum 50k data
Found 125 of ki data for polymerid = 49000265,49000267
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50240609(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]-SI-Ang-2 from AT1 receptor in Rattus norvegicus Sprague-Dawley (rat) liver membranes after 2 hrMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]-SI-Ang-2 from AT1 receptor in Rattus norvegicus Sprague-Dawley (rat) liver membranes after 2 hrMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50043280(4'-((1,4'-dimethyl-2'-propyl(2,6'-bi-1H-benzimidaz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM82077(Angiotensin II | CAS_11128-99-7 | NSC_439662)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50009718(2-Ethyl-5,7-dimethyl-3-[2'-(1H-tetrazol-5-yl)-biph...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50006909(2-Butyl-5-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  0.570nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50003154(2-{Propyl-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM82259(CAS_123856 | L-158,809 | NSC_123856)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50287290(CHEMBL34866 | KRH-594 | Potassium; 2-[5-ethyl-3-[2...)
Affinity DataKi:  1.02nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]Ang2 from AT1 receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50082568(2-({3-[4-(2-Azido-benzenesulfonylaminocarbonyl)-be...)
Affinity DataKi:  1.5nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50009338((S)-2-((S)-1-((S)-2-((S)-2-((S)-2-((S)-2-((S)-5-(d...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50003155(4-{Butyl-[2''-(2H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50161275(CHEMBL3787059)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]-Ang II from Angiotensin 2 type-1A receptor in rat vascular smooth muscle cells after 150 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50141059(CHEMBL289614 | L-162782 | N-Butyloxycarbonyl-4'-(2...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [125]Ang2 from AT1 receptor in rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50082567(2-({2-Butyl-3-[4-(2-chloro-benzenesulfonylaminocar...)
Affinity DataKi:  2.5nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50003158(2-Methyl-4-{propyl-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50161276(CHEMBL3786570)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]-Ang II from Angiotensin 2 type-1A receptor in rat vascular smooth muscle cells after 150 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50011977((E)-2-butyl-1-(p-carboxybenzyl)-alpha-2-thenylimid...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]Ang II from AT1 receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50049189(3-[4-(2-Ethyl-57-dimethyl-imidazo[45-b]pyridin-3-y...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [I125I]AngII form AT1 receptor in rat liver membrane incubated for 1.5 hrs by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50161277(CHEMBL3787050)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-Ang II from Angiotensin 2 type-1A receptor in rat vascular smooth muscle cells after 150 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50082570(2-[2-butyl-1-(4-carboxybenzyl)-1H-5-imidazolylmeth...)
Affinity DataKi:  12.1nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKi:  12.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303975(3'-(4-(2-(1H-Tetrazol-5-yl)ethyl)benzyl)-1,7'-dime...)
Affinity DataKi:  13.4nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]-Ang II from Angiotensin 2 type-1A receptor in rat vascular smooth muscle cells after 150 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50119657(8-Butyl-7-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50003156(4-{Butyl-[2''-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  15nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKi:  15nMAssay Description:Binding affinity against angiotensin II receptor from rat liver; n=8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50045358(2-Ethyl-4-{[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataKi:  21nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50082569(4-Azido-2-{[2-butyl-3-(4-carboxy-benzyl)-3H-imidaz...)
Affinity DataKi:  22nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50089990(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  25nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50368649(CHEMBL1202852)
Affinity DataKi:  68nMAssay Description:Binding affinity against angiotensin II receptor from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50119658(7-Butyl-8-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataKi:  80nMAssay Description:Displacement of [125I]Sar1,Ile8-Ang2 from AT1 receptor in Wistar rat hepatic membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50487564(CHEMBL2260199)
Affinity DataKi:  188nMAssay Description:Displacement of [125I]-SI-Ang-2 from AT1 receptor in Rattus norvegicus Sprague-Dawley (rat) liver membranes after 2 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50487559(CHEMBL2260198)
Affinity DataKi:  650nMAssay Description:Displacement of [125I]-SI-Ang-2 from AT1 receptor in Rattus norvegicus Sprague-Dawley (rat) liver membranes after 2 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303976(3'-(2-(4-(2-(1H-Tetrazol-5-yl)ethyl)phenoxy)ethyl)...)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50514581(CHEMBL1885579)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [125I]Ang II from AT1 receptor in rat SMC membranes incubated for 60 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303977(3-(4-(2-(1,7'-Dimethyl-2'-propyl-1H,3'H-2,5'-biben...)
Affinity DataKi:  2.23E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303979(CHEMBL571763 | Ethyl 3-(4-(2-(1,7'-Dimethyl-2'-pro...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303978(1-(4-(2-(1H-tetrazol-5-yl)ethyl)benzyl)-4-methyl-2...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50303980(1-(4-((1H-Tetrazol-5-yl)methoxy)benzyl)-4-methyl-2...)
Affinity DataKi:  5.06E+3nMAssay Description:Displacement of [125I]SI-Ang2 from AT1 receptor in Sprague-Dawley rat liver membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Xenopus tropicalis)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandPNGBDBM82273(CAS_167710-87-4 | RS 39604)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50094703(5-(3-Bromo-phenyl)-7-(6-morpholin-4-yl-pyridin-3-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM86694(N'-(3-Chloro-4-morpholinophenyl)-N-hydroxyform...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50030814(CHEMBL2086892)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Ang II from AT1 receptor in rat liver membranes after 2 hrs by gamma-counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50156173((1-((2'-(1H-tetrazol-5-yl)biphenyl-4-yl)methyl)-2-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-Ang II from AT1 receptor in rat liver membranes after 2 hrs by gamma-counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor A(RAT)
Shinshu University

Curated by PDSP Ki Database
LigandPNGBDBM50221297(CHEMBL239393 | N-butyloxycarbonyl-3-[4-(N,N-dimeth...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Ang 2 from AT1 receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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