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TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423968(CHEMBL2313377)
Affinity DataEC50:  640nMAssay Description:Positive allosteric modulation of rat muscarinic M2 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258723(7-chloro-1-(4-(trifluoromethyl)benzyl)indoline-2,3...)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258723(7-chloro-1-(4-(trifluoromethyl)benzyl)indoline-2,3...)
Affinity DataEC50:  2.84E+3nMAssay Description:Activation of rat muscarinic M2 receptor expressed in CHO cells co-expressing chimeric Gqi5 protein assessed as potentiation of acetylcholine-induced...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356969(CHEMBL1916226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356968(CHEMBL1916225)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356973(CHEMBL1916235)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356978(CHEMBL1916233)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356972(CHEMBL1916234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356977(CHEMBL1916232)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356971(CHEMBL1916228)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356974(CHEMBL1916229)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356970(CHEMBL1916227)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356976(CHEMBL1916231)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356975(CHEMBL1916230)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50023229(CHEMBL3329755)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat muscarinic acetylcholine receptor subtype 2 expressed in CHO cells co-transfected with chimeric Gqi5 by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207517(CHEMBL3915634)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356969(CHEMBL1916226)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207463(CHEMBL3963788)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207516(CHEMBL3942511)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M2 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50451549(CHEMBL4207737)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulator activity at rat M2 receptor expressed in CHO cells co-expressing Gqi5 assessed as maximal response to ACh by calcium mo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423967(CHEMBL2057417)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M2 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50263887(1-(1'-2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-be...)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50249403(CHEMBL4091821)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat M2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258439(cid_3008304 | CHEMBL523685 | VU0119498 | 1-(4-brom...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M2 expressed in CHO cells assessed as stimulation of calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M2 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43821(4-(2-benzamidoethylamino)-1-piperidinecarboxylic a...)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at rat muscarinic M2 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M2 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M2(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50615274(CHEMBL5283571)
Affinity DataEC50: >5.10E+4nMAssay Description:Agonist activity at rat M2 muscarinic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed