Compile Data Set for Download or QSAR
Report error Found 29 of ec50 for UniProtKB: P08911
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433574BDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.224nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433574BDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.225nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258656BDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258656BDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258656BDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50258656BDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433574BDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50433574BDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50023229BDBM50023229(CHEMBL3329755)
Affinity DataEC50:  610nMAssay Description:Activity at rat muscarinic acetylcholine receptor subtype 5 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356973BDBM50356973(CHEMBL1916235)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356977BDBM50356977(CHEMBL1916232)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356976BDBM50356976(CHEMBL1916231)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356972BDBM50356972(CHEMBL1916234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356978BDBM50356978(CHEMBL1916233)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356971BDBM50356971(CHEMBL1916228)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356970BDBM50356970(CHEMBL1916227)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356975BDBM50356975(CHEMBL1916230)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356974BDBM50356974(CHEMBL1916229)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356969BDBM50356969(CHEMBL1916226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356968BDBM50356968(CHEMBL1916225)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50249403BDBM50249403(CHEMBL4091821)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207516BDBM50207516(CHEMBL3942511)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50546065BDBM50546065(CHEMBL4795177)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207463BDBM50207463(CHEMBL3963788)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50207517BDBM50207517(CHEMBL3915634)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50423967BDBM50423967(CHEMBL2057417)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50423968BDBM50423968(CHEMBL2313377)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50356966BDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 43822BDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed