TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 21nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 43nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 220nMAssay Description:In vitro Binding affinity towards alpha-3 (PC12) nAChR was determinedMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 240nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 310nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 350nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 490nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 580nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 610nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 2.20E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 2.30E+3nMAssay Description:In vitro Binding affinity towards alpha-3 (PC12) nAChR was determinedMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 2.90E+3nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 3.16E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 5.01E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Affinity DataKi: 6.30E+3nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 7.20E+3nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Human)
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 9.06E+3nMAssay Description:Binding affinity to alpha3beta4alpha5 nAChR (unknown origin)More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-6/beta-2/beta-3(Human)
Targacept
Curated by ChEMBL
Targacept
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]epibatidine from human alpha6/alpha3beta2beta3 nAChR transfected in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
Sanofi-Synthelabo Research
Curated by PDSP Ki Database
Sanofi-Synthelabo Research
Curated by PDSP Ki Database














































