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Found 248 of ec50 for UniProtKB: A0A024R4H6
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100081(4-[[2-(4-fluorophenyl)-4-keto-1,2-dihydroquinazoli...)
Affinity DataEC50: >286nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM75191(2-[7-hydroxy-2-keto-4-methyl-8-[(veratrylamino)met...)
Affinity DataEC50: >858nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100095(2-Oxo-1,2-dihydro-benzo[cd]indole-6-sulfonic acid ...)
Affinity DataEC50:  1.84E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100052((Z)-3-(1,3-benzothiazol-2-yl)-N-(4-chlorobenzyl)-4...)
Affinity DataEC50:  2.56E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100194(3-(3,4-dimethylphenyl)-N-[(2-methoxy-1-naphthaleny...)
Affinity DataEC50: >2.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100179(1-[2-(2-Hydroxy-ethoxy)-ethylamino]-3-propyl-benzo...)
Affinity DataEC50: >2.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81149(MLS001213181 | N'-(10H-indolo[3,2-b]quinolin-2-yl)...)
Affinity DataEC50: >2.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100036(1'-acetyl-6-[2-(4-ethyl-1-piperazinyl)-2-oxoethoxy...)
Affinity DataEC50: >2.58E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100103(3-(4-methoxyphenyl)-8-[(2-methylpiperidin-1-yl)met...)
Affinity DataEC50: >2.58E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100127(MLS001162224 | SMR000670895 | cid_4989776)
Affinity DataEC50: >2.58E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100049(3-(3,5-dimethylphenoxy)-4-oxo-4H-chromen-7-yl prop...)
Affinity DataEC50:  3.19E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM51528(2-amino-1-(2-piperidinoethyl)pyrrolo[3,2-b]quinoxa...)
Affinity DataEC50:  3.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100100(3-Methyl-1-methylamino-benzo[4,5]imidazo[1,2-a]pyr...)
Affinity DataEC50:  3.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100163(2-[4-amino-5-(4-methoxyphenyl)-3-methylpyrazolo[3,...)
Affinity DataEC50:  4.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM51482(5-cyano-6-[[2-(ethoxycarbonylamino)-2-oxoethyl]thi...)
Affinity DataEC50:  4.56E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100118(2-(2-keto-3-phenyl-chromen-7-yl)oxypropionic acid ...)
Affinity DataEC50:  5.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100031(MLS000527663 | N-(2,3-dimethyl-6-quinoxalinyl)-1-p...)
Affinity DataEC50:  5.48E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100151((4-oxidanylidene-5,6,7,8-tetrahydro-3H-[1]benzothi...)
Affinity DataEC50:  6.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100070(7-(diethylamino)-3-(hydroxymethyl)-4-methyl-1-benz...)
Affinity DataEC50:  6.34E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM90096(MLS000578964 | SMR000198786 | butyl 3-(3-methylphe...)
Affinity DataEC50:  6.86E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50549(2-(5-methyl-2-furanyl)-4-quinolinecarboxylic acid ...)
Affinity DataEC50:  6.97E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100171(MLS002920943 | N-((2S,3R,12bS)-3-((S)-1-hydroxyeth...)
Affinity DataEC50:  7.44E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100162(3-[(3R,4S)-4-ethyl-5-(4-fluorophenyl)-2-phenyl-2-p...)
Affinity DataEC50:  7.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100143(MLS001035725 | N-[4-[2-(2-methoxyphenyl)ethanoylam...)
Affinity DataEC50:  7.57E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM82911(2-(2-furanyl)-6-(2-propan-2-yloxyethoxy)-1-benzopy...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100182(1-[2-methyl-1-(2-methylprop-2-enyl)-3-oxidanyliden...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100077(2-amino-5-chloro-benzoic acid [2-[(1,1-diketothiol...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100116(MLS001176569 | SMR000595898 | cid_4962774)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM46572((6E)-5-azanylidene-6-[(4-oxidanylidenechromen-3-yl...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100189(4-[7-(4-carbamoylphenyl)-1-(2-cyclopropyl-2-keto-e...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50016479((7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]qui...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100058(MLS000718244 | N-cyclopentyl-2-(4-fluorophenyl)-3-...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100146(1-[2-(4-butyl-2-keto-7-methyl-chromen-5-yl)oxyacet...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100185(MLS003124389 | SMR001285658 | [3-[6-(methylamino)-...)
Affinity DataEC50: >7.72E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100062(5-keto-8-methyl-N-(tetrahydrofurfuryl)-2-(tetrahyd...)
Affinity DataEC50:  7.79E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100164(MLS002582724 | N-[3-cyano-1-(2-furanylmethyl)-10-m...)
Affinity DataEC50:  7.95E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100019(4-[[3-cyano-6-methyl-4-(3-pyridinyl)-2-pyridinyl]t...)
Affinity DataEC50:  8.07E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100191(1-[1-(1H-benzimidazol-2-yl)ethyl]-3-(2-thienyl)qui...)
Affinity DataEC50:  8.14E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100186((2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-N-[5-(dimethyl...)
Affinity DataEC50:  8.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100087((4S)-6-amino-5-cyano-2-(2-keto-2-methoxy-ethyl)-4-...)
Affinity DataEC50:  8.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100045(6,7-dimethoxy-2-methyl-2,3-dihydro-1-benzothiopyra...)
Affinity DataEC50:  8.28E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100129(MLS001223360 | N-[4-[2-(2-chloranylphenoxy)ethanoy...)
Affinity DataEC50:  8.31E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100173(2-ethyl-3-(2-ethylbutyl)-9,10-dimethoxy-1,3,4,6,7,...)
Affinity DataEC50:  8.32E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100005(1-(9-methoxy-5H-pyrimid[5,4-b]indol-4-yl)isonipeco...)
Affinity DataEC50:  8.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100172(1-[(2S,3R,12bS)-3-[(1S)-1-hydroxyethyl]-4-keto-2,3...)
Affinity DataEC50:  8.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100074(MLS000419029 | N-(1,3-diketoisoindolin-5-yl)-4-pyr...)
Affinity DataEC50:  8.55E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100024(MLS000113735 | N-(2-thiophen-2-yl-3H-benzimidazol-...)
Affinity DataEC50:  8.78E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100165(2-[(1S,3R,12bS)-10-(2-furanyl)-4-oxo-1-[oxo(1-pipe...)
Affinity DataEC50:  8.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM100167(MLS002694422 | N-(2-fluoranthenyl)acetamide | N-fl...)
Affinity DataEC50:  8.84E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetKallikrein-7(Homo sapiens (Human))
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50241529(7-hydroxy-6-methoxy-3-(4-methoxyphenyl)-4H-chromen...)
Affinity DataEC50:  9.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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