Compile Data Set for Download or QSAR
Report error Found 3 of affinity data for UniProtKB/TrEMBL: Q96NY9
TargetCrossover junction endonuclease MUS81(Homo sapiens)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50618708(CHEMBL4071130)
Affinity DataKd:  6.10nMAssay Description:Binding affinity to human GST-tagged MUS81-ECE2 expressed in Escherichia coli BL21(DE3)Rosetta2 cells assessed as dissociation constant by Surface pl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCrossover junction endonuclease MUS81(Homo sapiens)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50323460(N'-(3,4-dihydroxybenzylidene)-3-hydroxy-2-naphthoh...)
Affinity DataKd:  4.20nMAssay Description:Binding affinity to human GST-tagged MUS81-ECE2 expressed in Escherichia coli BL21(DE3)Rosetta2 cells assessed as dissociation constant by Surface pl...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetCrossover junction endonuclease MUS81(Homo sapiens)
Fuzhou University

Curated by ChEMBL
LigandPNGBDBM50618708(CHEMBL4071130)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human GST-tagged MUS81-ECE2 expressed in Escherichia coli BL21(DE3)Rosetta2 cells incubated for 15 mins by FRET based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed