TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 8.17E+3nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair
TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 82nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair
TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair
TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 2.70E+3nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair
TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: >2.30E+4nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair
TargetRyanodine receptor 2(Homo sapiens)
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Max Planck Institute for Multidisciplinary Sciences
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Modulator activity at wild type RyR2 (unknown origin) expressed in HEK293T co-expressed with R-CEPIA1er assessed as decrease in RyR2-mediated calcium...More data for this Ligand-Target Pair