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Found 14 of ec50 data for polymerid = 50001773
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50426567(BMS-204352 | FLINDOKALNER | MaxiPost)
Affinity DataEC50:  352nMAssay Description:Positive modulation of Kca 1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128974(2-Azepan-1-yl-1H-pyrrolo[3,2-b]pyridine-3-carbonit...)
Affinity DataEC50:  3.34E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128985(2-Morpholin-4-yl-1H-pyrrolo[3,2-b]pyridine-3-carbo...)
Affinity DataEC50:  3.86E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128979(2-(3-Aza-bicyclo[3.2.2]non-3-yl)-1H-pyrrolo[3,2-b]...)
Affinity DataEC50:  4.43E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128975(2-((S)-3-Hydroxy-piperidin-1-yl)-1H-pyrrolo[3,2-b]...)
Affinity DataEC50:  5.07E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128973(2-Dimethylamino-1H-pyrrolo[3,2-b]pyridine-3-carbon...)
Affinity DataEC50:  5.13E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128978(2-Imidazol-1-yl-1H-pyrrolo[3,2-b]pyridine-3-carbon...)
Affinity DataEC50:  5.86E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128984(2-[(2-Dimethylamino-ethyl)-methyl-amino]-1H-pyrrol...)
Affinity DataEC50:  6.75E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128982(2-Diethylamino-1H-pyrrolo[3,2-b]pyridine-3-carboni...)
Affinity DataEC50:  6.94E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128980(2-Pyrrolidin-1-yl-1H-pyrrolo[3,2-b]pyridine-3-carb...)
Affinity DataEC50:  8.12E+3nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128977(2-Hydroxy-1H-pyrrolo[3,2-b]pyridine-3-carbonitrile...)
Affinity DataEC50:  1.34E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128976(2-(4-Hydroxy-piperidin-1-yl)-1H-pyrrolo[3,2-b]pyri...)
Affinity DataEC50:  1.51E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50128981(1-(3-Cyano-1H-pyrrolo[3,2-b]pyridin-2-yl)-piperidi...)
Affinity DataEC50:  1.70E+4nMAssay Description:[86Rb+] efflux induced by BKca alpha subunits expressed in HEK293 cells at 10 microMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalcium-activated potassium channel subunit alpha-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50593373(CHEMBL5182581)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of Maxi-K channel (unknown origin) by thallium flux assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed