Compile Data Set for Download or QSAR
Report error Found 26 of ki for UniProtKB: Q64737
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50005868(CHEMBL38902 | 2-{4-[(2-Amino-4-oxo-3,4,5,6,7,8-hex...)
Affinity DataKi:  47nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM22590(5,10-dideazatetrahydrofolic acid | DDF | (2S)-2-[(...)
Affinity DataKi:  60nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024475(2-{4-[(2-Amino-4-oxo-1,4,5,6,7,8-hexahydro-quinazo...)
Affinity DataKi:  65nMAssay Description:In vitro inhibition of mouse GAR transformylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50367875(CHEMBL607957)
Affinity DataKi: >100nMAssay Description:Compound was tested for inhibition constant against GAR TFase in miceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM22590(5,10-dideazatetrahydrofolic acid | DDF | (2S)-2-[(...)
Affinity DataKi:  120nMAssay Description:Tested for the inhibition of trifunctional Glycinamide ribonucleotide formyltransferase isolated from murine L1210 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50003896((DDATHF) 5,10-Dideazatetrahydrofolic acid2-{4-[2-(...)
Affinity DataKi:  120nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50291133(2-{(S)-4-[2-(8-Amino-6-oxo-2,3,4,5,6,7-hexahydro-1...)
Affinity DataKi:  147nMAssay Description:Tested in vitro for its inhibition of trifunctional glycinamide ribonucleotide formyltransferase (GARFT) isolated from murine L1210 leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50005865(CHEMBL417696 | 2-{4-[(2-Amino-4-oxo-3,4,5,6,7,8-he...)
Affinity DataKi:  190nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50073753((R)-2-({5-[2-(2,4-Diamino-5,6,7,8-tetrahydro-pyrid...)
Affinity DataKi:  710nMAssay Description:Inhibitory activity against murine glycinamide ribonucleotide formyltransferase (GARFT) enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024464(2-{4-[Acetyl-(2-amino-4-oxo-3,4-dihydro-quinazolin...)
Affinity DataKi:  1.30E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50002471(CHEMBL289923 | 5-Amino-2-{4-[(2-amino-4-oxo-2,3,4,...)
Affinity DataKi:  1.40E+3nMAssay Description:potent inhibitor of GAR Tfase obtained from porcineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50006906(CHEMBL23977 | 2-{4-[(2-Amino-4-oxo-3,4-dihydro-qui...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024465(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50002471(CHEMBL289923 | 5-Amino-2-{4-[(2-amino-4-oxo-2,3,4,...)
Affinity DataKi:  3.70E+3nMAssay Description:In vitro inhibition of glycinamide ribonucleotide formyltransferase from L1210 murine leukemia cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024468(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50008294(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024466(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024467(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50073752(LY-335580 | (R)-2-({5-[2-(2,4-Diamino-5,6,7,8-tetr...)
Affinity DataKi:  9.20E+3nMAssay Description:Inhibitory activity against murine glycinamide ribonucleotide formyltransferase (GARFT) enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024462(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50017876(CHEMBL22632 | 2-{4-[(2-Amino-4-oxo-3,4-dihydro-qui...)
Affinity DataKi:  1.60E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024461(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024463(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  1.90E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50281128((S)-2-{4-[2-(4-Oxo-3,4,5,6,7,8-hexahydro-pyrido[2,...)
Affinity DataKi:  2.70E+4nMAssay Description:Tested for the inhibition against the human dihydrofolate reductaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50024469(2-{4-[(2-Amino-4-oxo-3,4-dihydro-quinazolin-6-ylme...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of GAR transformylase isolated from the murine lymphoma cell line L5178YMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrifunctional purine biosynthetic protein adenosine-3(Mouse)
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50073754((R)-2-{4-[2-(2,4-Diamino-5,6,7,8-tetrahydro-pyrido...)
Affinity DataKi:  5.60E+4nMAssay Description:Inhibitory activity against murine glycinamide ribonucleotide formyltransferase (GARFT) enzymeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed