Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for UniProtKB: P02751
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Ariad Pharmaceuticals

LigandPNGBDBM50244569(AP24283 | CHEMBL510893 | N-(4-(dimethylphosphoryl)...)
Affinity DataIC50: <0.5nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Ariad Pharmaceuticals

LigandPNGBDBM50244430(9-(2,6-dimethylstyryl)-N-(4-(dimethylphosphoryl)ph...)
Affinity DataIC50:  9.10nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Ariad Pharmaceuticals

LigandPNGBDBM50244527(9-(2-(1H-indazol-4-yl)vinyl)-N-(4-(dimethylphospho...)
Affinity DataIC50:  17nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Fibronectin (1)(Homo sapiens (Human))
Ariad Pharmaceuticals

LigandPNGBDBM50244526(9-(2-(1H-indol-4-yl)vinyl)-N-(4-(dimethylphosphory...)
Affinity DataIC50:  198nMAssay Description:In vitro kinase assay using Abl, Abl T315I or Src kinase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed