Compile Data Set for Download or QSAR
Report error Found 36 of ki for UniProtKB: Q58F21
TargetBromodomain testis-specific protein [251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.0660nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137,251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0760nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.0860nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.290nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137,251-382](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205431BDBM205431((6S+2S)-PEG1 (7))
Affinity DataKi:  0.420nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein [21-137](Human)
Dana-Farber Cancer Institute

LigandChemical structure of BindingDB Monomer ID 205453BDBM205453(MTI (35))
Affinity DataKi:  0.560nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2016
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457489BDBM50457489(CHEMBL4208129)
Affinity DataKi:  0.690nMAssay Description:Binding affinity to BRDT bromodomain 1 to 2 (N21to P380 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by br...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 439497BDBM439497(US10633379, Example 82 | US10633379, Example 35)
Affinity DataKi:  1nMAssay Description:Inhibition of BRDT BD2 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 220447BDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to BRDT BD1 to BD2 (N21 to P380 residues) (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457496BDBM50457496(CHEMBL4217457)
Affinity DataKi:  4.20nMAssay Description:Binding affinity to BRDT bromodomain 1 to 2 (N21to P380 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by br...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50457495BDBM50457495(CHEMBL4215988)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to BRDT bromodomain 1 to 2 (N21to P380 amino acids) (unknown origin) using Alexa647-labeled BET-inhibitor as fluorescent probe by br...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260093BDBM50260093(CHEMBL4078100)
Affinity DataKi:  100nMAssay Description:Inhibition of human BRDT bromodomain 1 expressed in bacterial expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 342597BDBM342597(N-[3-(3-methyl-4-oxo-4,5,6,7-tetrahydro-2H-isoindo...)
Affinity DataKi:  110nMAssay Description:Binding affinity to BRDT BD1-BD2 (N21 to P380 residues) (unknown origin) after 1 hr by Alexa-647-conjugated probe based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158624BDBM50158624(CHEMBL3786012)
Affinity DataKi:  140nMAssay Description:Binding affinity to BRDT BD1-BD2 (N21 to P380 residues) (unknown origin) after 1 hr by Alexa-647-conjugated probe based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239566BDBM50239566(CHEMBL4103140)
Affinity DataKi:  200nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239567BDBM50239567(CHEMBL4085204)
Affinity DataKi:  200nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239568BDBM50239568(CHEMBL4092949)
Affinity DataKi:  220nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239565BDBM50239565(CHEMBL4065286)
Affinity DataKi:  230nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50256397BDBM50256397(CHEMBL4088466)
Affinity DataKi:  490nMAssay Description:Binding affinity to BRDT BD1-BD2 (N21 to P380 residues) (unknown origin) after 1 hr by Alexa-647-conjugated probe based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50260093BDBM50260093(CHEMBL4078100)
Affinity DataKi:  501nMAssay Description:Inhibition of human BRDT bromodomain 2 expressed in bacterial expression systemMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239562BDBM50239562(CHEMBL4104179)
Affinity DataKi:  690nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239586BDBM50239586(CHEMBL4072799)
Affinity DataKi:  850nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 439497BDBM439497(US10633379, Example 82 | US10633379, Example 35)
Affinity DataKi:  917nMAssay Description:Inhibition of BRDT BD1 (unknown origin) after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239588BDBM50239588(CHEMBL4077905)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239585BDBM50239585(CHEMBL4094028)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239571BDBM50239571(CHEMBL4088746)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239574BDBM50239574(CHEMBL4094424)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239577BDBM50239577(CHEMBL4064204)
Affinity DataKi:  5.60E+3nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239576BDBM50239576(CHEMBL4093510)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239578BDBM50239578(CHEMBL4085767)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239573BDBM50239573(CHEMBL4102160)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239587BDBM50239587(CHEMBL4067951)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239572BDBM50239572(CHEMBL4060512)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239570BDBM50239570(CHEMBL4066490)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239575BDBM50239575(CHEMBL4066935)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed
TargetBromodomain testis-specific protein(Human)
Abbvie

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50239569BDBM50239569(CHEMBL4086263)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of BI-BODIPY binding to BRDT bromodomain 1 (29 to 134 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) by fluorescence a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details Article
PubMed