Compile Data Set for Download or QSAR
maximum 50k data
Found 36 of ic50 for UniProtKB: A0A024R5S4
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50591324(CHEMBL5185273)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of N-terminal His-6 tagged USP8 (734 to 1110 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells measured after 3 hr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50591322(CHEMBL5196686)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of N-terminal His-6 tagged USP8 (734 to 1110 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells measured after 3 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50591323(CHEMBL5173239)
Affinity DataIC50:  2nMAssay Description:Inhibition of N-terminal His-6 tagged USP8 (734 to 1110 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells measured after 3 hr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50591321(CHEMBL5172138)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of N-terminal His-6 tagged USP8 (734 to 1110 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells measured after 3 hr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50436151(CHEMBL2398212)
Affinity DataIC50:  96nMAssay Description:Inhibition of human full-length His-tagged USP8 expressed baculovirus infected insect cells using Ub-AMC as substrate by fluorescence spectroscopic a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597448(CHEMBL5180195)
Affinity DataIC50:  280nMAssay Description:Inhibition of human full length USP8 overexpressed in baculovirus-infected insect cells using ubiquitin-C-terminal 7-amido-4-methylcoumarin as substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597449(CHEMBL5170305)
Affinity DataIC50:  290nMAssay Description:Inhibition of human full length USP8 overexpressed in baculovirus-infected insect cells using ubiquitin-C-terminal 7-amido-4-methylcoumarin as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597451(CHEMBL5202404)
Affinity DataIC50:  560nMAssay Description:Inhibition of human full length USP8 overexpressed in baculovirus-infected insect cells using ubiquitin-C-terminal 7-amido-4-methylcoumarin as substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597450(CHEMBL5208383)
Affinity DataIC50:  850nMAssay Description:Inhibition of human full length USP8 overexpressed in baculovirus-infected insect cells using ubiquitin-C-terminal 7-amido-4-methylcoumarin as substr...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597468(CHEMBL5184337)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597448(CHEMBL5180195)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597463(CHEMBL5176518)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597452(CHEMBL5171659)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells using ubiquitin-rhodamine -110 as substrate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597469(CHEMBL5197403)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597467(CHEMBL5206972)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50548233(CHEMBL4756029)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of USP8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50538571(CHEMBL4635160)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human USP8 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine110-glycine u...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597465(CHEMBL5205340)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597457(CHEMBL4469440)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597455(CHEMBL5206674)
Affinity DataIC50:  1.62E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597464(CHEMBL5181521)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597462(CHEMBL4536844)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597456(CHEMBL5198716)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597458(CHEMBL4591454)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597466(CHEMBL5170419)
Affinity DataIC50:  2.35E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597454(CHEMBL5175647)
Affinity DataIC50:  2.45E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597453(CHEMBL4567355)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50436152(SPONGIACIDIN C)
Affinity DataIC50: >3.16E+4nMAssay Description:Inhibition of core catalytic domain of USP8 (unknown origin) using ubiquitin-Rh110 as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597459(CHEMBL5170083)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597461(CHEMBL5180339)
Affinity DataIC50:  4.37E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50597460(CHEMBL5185694)
Affinity DataIC50:  4.52E+4nMAssay Description:Inhibition of N-terminal His6-tagged USP8 (unknown origin) catalytic domain (734 to 1110 residues) expressed in Escherichia coli BL21 (DE3) cells ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50007788(CHEMBL3233809 | med.21724, Compound 167)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human USP8 using Ub-rhodamine 110 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50007790(CHEMBL3233814 | med.21724, Compound 169)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human USP8 using Ub-rhodamine 110 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50007791(CHEMBL3233815 | med.21724, Compound 168)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human USP8 using Ub-rhodamine 110 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50007789(CHEMBL1173044 | GRL-0667 | N-(2H-1,3-benzodioxol-5...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human USP8 using Ub-rhodamine 110 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 8(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50271098(CHEMBL4129140)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of USP8 (unknown origin) expressed in baculovirus infected Sf9 cells using Ub-AMC as substrate preincubated for 30 mins followed by substr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed