Compile Data Set for Download or QSAR
maximum 50k data
Found 106 of ec50 for UniProtKB: A0A1L4FMK7
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105981(CHEMBL3598052)
Affinity DataEC50:  600nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106011(CHEMBL3598077)
Affinity DataEC50:  800nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105930(CHEMBL3598049)
Affinity DataEC50:  800nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105925(CHEMBL3598044)
Affinity DataEC50:  900nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105929(CHEMBL3598048)
Affinity DataEC50:  1.00E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50108881(CHEMBL3596591)
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at human ROR-beta transfected in HEK293T cells by Gal4 luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105932(CHEMBL3598050)
Affinity DataEC50:  1.10E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50050087(CHEMBL3317840 | US9216988, 50)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106008(CHEMBL3598075)
Affinity DataEC50:  1.30E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105928(CHEMBL3598047)
Affinity DataEC50:  1.30E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106002(CHEMBL3598070)
Affinity DataEC50:  1.30E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105982(CHEMBL3598053)
Affinity DataEC50:  1.50E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105933(CHEMBL3598051)
Affinity DataEC50:  1.70E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106007(CHEMBL3598074)
Affinity DataEC50:  1.80E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)
Affinity DataEC50:  1.93E+3nMAssay Description:Inverse agonist activity at Gal4 DNA binding domain-tagged human RORbeta expressed in HEK293T cells assessed as effect on receptor-mediated transcrip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50452782(CHEMBL4210791)
Affinity DataEC50: >2.00E+3nMAssay Description:Inverse agonist activity at Gal4-tagged human RORbeta ligand binding domain expressed in human Jurkat cells by native IL17 promoter driven luciferase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataEC50:  2.20E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106009(CHEMBL3598076)
Affinity DataEC50:  2.30E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012130(CHEMBL3263710)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012130(CHEMBL3263710)
Affinity DataEC50:  2.50E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012130(CHEMBL3263710)
Affinity DataEC50:  2.50E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50090086(CHEMBL3581533 | US9216988, 92)
Affinity DataEC50:  2.70E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50035885(CHEMBL3361064)
Affinity DataEC50: >3.10E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50044160(CHEMBL3314003)
Affinity DataEC50:  3.40E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012124(CHEMBL3263714)
Affinity DataEC50:  3.70E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50035907(CHEMBL3361050)
Affinity DataEC50:  3.80E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50426729(CHEMBL2326845)
Affinity DataEC50:  4.00E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50452782(CHEMBL4210791)
Affinity DataEC50: >4.00E+3nMAssay Description:Agonist activity at Gal4-tagged human RORbeta ligand binding domain expressed in human Jurkat cells by native IL17 promoter driven luciferase reporte...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50121988(CHEMBL3617309)
Affinity DataEC50:  4.10E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50444335(CHEMBL3094367)
Affinity DataEC50:  5.00E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012122(CHEMBL3263695)
Affinity DataEC50:  5.00E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50536791(CHEMBL4579711)
Affinity DataEC50:  5.40E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as activation of basal transcriptional activity by dual-glo luci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50121938(CHEMBL3617295)
Affinity DataEC50:  5.40E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at RoRb (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 NR reporter cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50444333(CHEMBL3094369)
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at RoRb (unknown origin) expressed in HEK293 cells assessed as transcriptional activity by GAL4 NR reporter cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50444333(CHEMBL3094369)
Affinity DataEC50:  6.00E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM19993(CHEMBL62136 | N-[4-(1,1,1,3,3,3-hexafluoro-2-hydro...)
Affinity DataEC50:  6.00E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50105984(CHEMBL3598054)
Affinity DataEC50:  6.20E+3nMAssay Description:Inverse agonist activity at RORbeta (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50536796(CHEMBL4560046)
Affinity DataEC50:  6.80E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as activation of basal transcriptional activity by dual-glo luci...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50121939(CHEMBL3617297)
Affinity DataEC50:  7.90E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293 cells assessed as suppression of basal transcriptional activity after 20 hrs by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50035918(CHEMBL3361061)
Affinity DataEC50: >8.00E+3nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50545540(CHEMBL4644223)
Affinity DataEC50:  8.30E+3nMAssay Description:Agonist activity at Gal4-fused RORbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50548025(CHEMBL4782326)
Affinity DataEC50:  8.40E+3nMAssay Description:Inverse agonist activity at Gal4-fused RORbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50012126(CHEMBL3263716)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORb expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50035908(CHEMBL3361051)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50035915(CHEMBL3361058)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50050083(CHEMBL3317833 | US9216988, 101)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50050086(CHEMBL3317836 | US9216988, 55)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50050117(CHEMBL3317843 | US9216988, 54)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs by dual-g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor ROR-beta(Homo sapiens (Human))
Biogen

Curated by ChEMBL
LigandPNGBDBM50106286(CHEMBL3598141 | US9550771, Example 27)
Affinity DataEC50: >1.00E+4nMAssay Description:Inverse agonist activity at GAL4-fused human RORb expressed in HEK293T cells assessed as suppression of basal transcriptional activity after 20 hrs b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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