Compile Data Set for Download or QSAR
maximum 50k data
Found 176 of ic50 for UniProtKB: P09217
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50468260(CHEMBL4282837)
Affinity DataIC50:  1nMAssay Description:Inhibition of rat brain PKC using RGFR derived peptide substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469649(CHEMBL283259)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469642(CHEMBL282805)
Affinity DataIC50:  2.40nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469642(CHEMBL282805)
Affinity DataIC50:  2.40nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  3nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50108296(CHEMBL289772 | Indolocarbazole analogue)
Affinity DataIC50:  3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469644(CHEMBL281448)
Affinity DataIC50:  5nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  6nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469655(CHEMBL26872)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  9nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469652(CHEMBL285613)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  10nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469643(CHEMBL284632)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469641(CHEMBL283903)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469640(CHEMBL26817)
Affinity DataIC50:  15nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50478518(CHEMBL514017)
Affinity DataIC50:  17nMAssay Description:Displacement of [3H]PDBu from rat brain membrane PKCMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469645(CHEMBL26074)
Affinity DataIC50:  17nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469646(CHEMBL27387)
Affinity DataIC50:  19nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469639(CHEMBL282298)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469650(CHEMBL283399)
Affinity DataIC50:  20nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM3033(3-{23-methyl-14-oxo-3,13,23-triazahexacyclo[14.7.0...)
Affinity DataIC50:  20nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469647(CHEMBL283930)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469653(CHEMBL282612)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280871(12-(3-azidopropyl)-13-methyl-6,7,12,13-tetrahydro-...)
Affinity DataIC50:  25nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50:  27nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50:  32nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50478561(CHEBI:69599 | Methylpendolmycin)
Affinity DataIC50:  35.2nMAssay Description:Displacement of radiolabeled PDBU from PKC in rat forebrainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50241867(((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...)
Affinity DataIC50:  68nMAssay Description:Displacement of [3H]PDBu from rat brain PKC by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50:  75nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469654(CHEMBL28202)
Affinity DataIC50:  86nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469651(CHEMBL26996)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50:  99nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)
Affinity DataIC50:  100nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280875(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50:  110nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50469648(CHEMBL26936)
Affinity DataIC50:  145nMAssay Description:In vitro inhibition of protein kinase C from rat brain.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50:  200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128287(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-methyl-piperidi...)
Affinity DataIC50:  200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128280(3-[1-(1-Ethyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128282(3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50108291(CHEMBL36891 | Indolocarbazole analogue)
Affinity DataIC50:  222nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM6760((+)-K-252a | CHEMBL281948 | K-252a | methyl (15S,1...)
Affinity DataIC50:  250nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128286(3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...)
Affinity DataIC50:  250nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128290(3-[1-(1-Cyclopropylmethyl-piperidin-4-yl)-1H-indol...)
Affinity DataIC50:  300nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM50217039(CHEMBL420938)
Affinity DataIC50:  300nMAssay Description:Inhibition of protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Pak Research Center

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  300nMAssay Description:Inhibition of PKC in rat RBL2H3 cells assessed as inhibition of mouse anti-DNP IgE-stimulated beta-hexosaminidase release preincubated for 15 mins fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128281(18-dimethylaminomethyl-(18S)-17-oxa-4,14,21-triaza...)
Affinity DataIC50:  320nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50108299(CHEMBL288229 | Indolocarbazole analogue)
Affinity DataIC50:  400nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50128288(3-(1-Methyl-1H-indol-3-yl)-4-(1-piperidin-4-yl-1H-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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