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TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50303364(1-(4-((Benzo[d]oxazol-2-ylthio)methyl)phenyl)-3,3-...)
Affinity DataKd:  3nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50303363(2-(4-(3,3-Diethyl-2,4-dioxoazetidin-1-yl)benzylthi...)
Affinity DataKd:  9.5nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50235614(3,3-diethyl-1-(4-tolyl)azetidine-2,4-dione | 3,3-d...)
Affinity DataKd:  48.2nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50235612(1-(4-chlorophenyl)-3,3-diethylazetidine-2,4-dione ...)
Affinity DataKd:  57.9nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50303365(1-(2-((Benzo[d]oxazol-2-ylthio)methyl)phenyl)-3,3-...)
Affinity DataKd:  205nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50303362(1-(2-((Benzo[d]thiazol-2-ylthio)methyl)phenyl)-3,3...)
Affinity DataKd:  283nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50303367(1-(2-((5-Phenyl-1,3,4-oxadiazol-2-ylthio)methyl)ph...)
Affinity DataKd:  353nMAssay Description:Inhibition of human leukocyte elastase after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2010
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50084227(2-Diethylamino-5-methyl-4-oxo-4H-thieno[2,3-d][1,3...)
Affinity DataKd:  620nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
University of Lisbon

Curated by ChEMBL
LigandPNGBDBM50084228(2-(diethylamino)-5-methyl-4H-thieno[2,3-d][1,3]oxa...)
Affinity DataKd:  5.50E+3nMAssay Description:Inhibitory activity against human leukocyte elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed