Compile Data Set for Download or QSAR
maximum 50k data
Found 9699 of ic50 for UniProtKB: P24941
LigandPNGBDBM50378288(CHEMBL567434)
Affinity DataIC50:  0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378304(CHEMBL568080)
Affinity DataIC50: <0.0300nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378319(CHEMBL568303)
Affinity DataIC50: <0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378289(CHEMBL565705)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378290(CHEMBL568310)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378291(CHEMBL568302)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378305(CHEMBL583417)
Affinity DataIC50: <0.0400nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378292(CHEMBL566106)
Affinity DataIC50:  0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50003691(CHEMBL567624)
Affinity DataIC50: <0.0500nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50003691(CHEMBL567624)
Affinity DataIC50: <0.0500nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378293(CHEMBL566550)
Affinity DataIC50:  0.0600nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378292(CHEMBL566106)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378294(CHEMBL566972)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378295(CHEMBL565490)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378290(CHEMBL568310)
Affinity DataIC50:  0.0800nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378288(CHEMBL567434)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378299(CHEMBL568079)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378298(CHEMBL583421)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378296(CHEMBL568510)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378297(CHEMBL566105)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378305(CHEMBL583417)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378304(CHEMBL568080)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378303(CHEMBL567208)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378302(CHEMBL583615)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378301(CHEMBL568311)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378289(CHEMBL565705)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378297(CHEMBL566105)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378300(CHEMBL565930)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378212(CHEMBL575450)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378306(CHEMBL567647)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378293(CHEMBL566550)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378298(CHEMBL583421)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378307(CHEMBL566329)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM601933(4-((6'-hydroxy-8'-oxo-7',8'-dihydro-6'H- spiro[cyc...)
Affinity DataIC50:  0.160nMAssay Description:Selected compounds disclosed herein were tested in kinase assays by Nanosyn (Santa Clara, Calif.) to determine their inhibitory effect on these CDKs....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
LigandPNGBDBM50378312(CHEMBL578664)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378313(CHEMBL567626)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378302(CHEMBL583615)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378314(CHEMBL578256)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378303(CHEMBL567208)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378311(CHEMBL568301)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378310(CHEMBL566971)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50378309(CHEMBL568093)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of Cdk2/cyclinEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM6878(1-Acyl-1H-[1,2,4]triazole-3,5-diamine Analogue 3n ...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of GST-tagged CDK2/cyclin A2 (unknown origin) expressed in Escherichia coli using histone H1 as substrate in presence of [gamma-33P]-ATP b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM642762(N-(1-(cyclopropylsulfonyl)piperidin-4-yl)-1-isopro...)
Affinity DataIC50:  0.200nMAssay Description:Assay of Kinase Activity The inhibitory effect of compounds against the kinase CDK4/cyclin D3 was detected by Caliper Mobility Shift Assay method. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM642760(1-isopropyl-N-(1-(methylsulfonyl)piperidin-4-yl)-1...)
Affinity DataIC50:  0.200nMAssay Description:Assay of Kinase Activity The inhibitory effect of compounds against the kinase CDK4/cyclin D3 was detected by Caliper Mobility Shift Assay method. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM642778(US20230416271, Compound II.32)
Affinity DataIC50:  0.200nMAssay Description:Assay of Kinase Activity The inhibitory effect of compounds against the kinase CDK4/cyclin D3 was detected by Caliper Mobility Shift Assay method. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM642777(1-isopropyl-N-(1-(methylsulfonyl)piperidin-4-yl)-4...)
Affinity DataIC50:  0.200nMAssay Description:Assay of Kinase Activity The inhibitory effect of compounds against the kinase CDK4/cyclin D3 was detected by Caliper Mobility Shift Assay method. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM642775(N-(1-(cyclopropylsulfonyl)piperidin-4-yl)-4-(diflu...)
Affinity DataIC50:  0.200nMAssay Description:Assay of Kinase Activity The inhibitory effect of compounds against the kinase CDK4/cyclin D3 was detected by Caliper Mobility Shift Assay method. Th...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50378300(CHEMBL565930)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant Cdk2/cyclinAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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