Compile Data Set for Download or QSAR
Report error Found 13 of ki data for polymerid = 7885
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50060417BDBM50060417(CHEMBL297784 | SB 206553 | SB-206553 | 5-Methyl-3,...)
Affinity DataKi:  10nMAssay Description:Binding affinity analysed on 5-HT 2C in human clone using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50017721BDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  11nMAssay Description:Binding affinity to 5-hydroxytryptamine 2C receptor using [3H]Mesulergine as radioligand in stably transfected NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 35920BDBM35920(CHEMBL47482 | 9-(Aminomethyl)-9,10-dihydroanthrace...)
Affinity DataKi:  43nMAssay Description:Binding affinity to 5-hydroxytryptamine 2C receptor using [3H]Mesulergine as radioligand in stably transfected NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82272BDBM82272(SB 200646 | SB200646a)
Affinity DataKi:  138nMAssay Description:Binding affinity analysed on 5-HT 2C in rat stomach fundusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010859BDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi:  160nMAssay Description:Binding affininity of the compound to 5-hydroxytryptamine 2C receptor using [3H]-Mesulergine as radioligand in stably transfected NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186969BDBM186969(US9079895, 32s)
Affinity DataKi:  1.11E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 84991BDBM84991(CAS_3277600 | NSC_3277600 | SB204741)
Affinity DataKi:  1.51E+3nMAssay Description:Binding affinity analysed on 5-HT 2C in human clone using [3H]mesulergine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186935BDBM186935(US9079895, 23s)
Affinity DataKi:  3.39E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186937BDBM186937(US9079895, 25s)
Affinity DataKi:  3.76E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186968BDBM186968(US9079895, 70)
Affinity DataKi:  6.37E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 186927BDBM186927(US9079895, 19s)
Affinity DataKi:  6.74E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
US Patent

Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50013515BDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity analysed towards 5-HT 2C in rat stomach fundusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Mouse)
Eli Lilly

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 85098BDBM85098(N-[5-[5-(2,4-Dioxo-1,3,8-triazaspiro[4.5]decan-8-y...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2012
Entry Details Article
PubMed