Compile Data Set for Download or QSAR
Report error Found 17 of kd for UniProtKB: P18825
TargetAlpha-2C adrenergic receptor(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50621980(ORM-13070 C-11 | 11c-orm-13070 | Orm-13070 c-11 | ...)
Affinity DataKd:  3.80nMAssay Description:Binding affinity to alpha2C receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  2.30E+3nMAssay Description:Dissociation constant in high affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  2.30E+3nMAssay Description:Dissociation constant in high affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  2.50E+4nMAssay Description:Dissociation constant in high affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  2.50E+4nMAssay Description:Dissociation constant in high affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  4.70E+4nMAssay Description:Dissociation constant in high affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  4.70E+4nMAssay Description:Dissociation constant in high affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  1.50E+5nMAssay Description:Dissociation constant in low affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  1.50E+5nMAssay Description:Dissociation constant in low affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  3.30E+5nMAssay Description:Dissociation constant in high affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  3.30E+5nMAssay Description:Dissociation constant in high affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  6.40E+5nMAssay Description:Dissociation constant in low affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  6.40E+5nMAssay Description:Dissociation constant in low affinity sites where the binding is in 50 mM phosphate buffer for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  2.50E+6nMAssay Description:Dissociation constant in low affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50027058((1S,2S,4aR,13bS,14aS)-2-Hydroxy-1,2,3,4,4a,5,7,8,1...)
Affinity DataKd:  2.50E+6nMAssay Description:Dissociation constant in low affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  5.40E+6nMAssay Description:Dissociation constant in low affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details

LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKd:  5.40E+6nMAssay Description:Dissociation constant in low affinity sites where the binding is in acetonitrile/acetic acid for Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2018
Entry Details