Compile Data Set for Download or QSAR
Report error Found 5 of ec50 for UniProtKB: P11275
LigandPNGBDBM6862(6-fluoro-3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0...)
Affinity DataIC50: 92nM EC50:  40nMT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]A...More data for this Ligand-Target Pair
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Date in BDB:
12/21/2005
Entry Details Article
PubMed
LigandPNGBDBM6859(7-bromo-3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^...)
Affinity DataIC50: 1.25E+3nM EC50:  70nMT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2005
Entry Details Article
PubMed
LigandPNGBDBM6860(6-bromo-3,13,23-triazahexacyclo[14.7.0.0^{2,10}.0^...)
Affinity DataIC50: 1.24E+4nM EC50:  70nMT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2005
Entry Details Article
PubMed
LigandPNGBDBM6768(indolocarbazole deriv. 4(f) | 20-bromo-3-methyl-3,...)
Affinity DataIC50: 174nM EC50:  80nMT: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]A...More data for this Ligand-Target Pair
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Date in BDB:
12/21/2005
Entry Details Article
PubMed
LigandPNGBDBM292485(US10100058, Example 141 | (S)-N-(2-(diethylamino)p...)
Affinity DataEC50:  120nMAssay Description:Inhibition of CaMK2alpha/beta in neonatal rat cortical neurons assessed as phospholamban phosphorylation after 4 hrs by Hoechst 33342 fluorescence-ba...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2020
Entry Details Article
PubMed