Compile Data Set for Download or QSAR
maximum 50k data
Found 14 of ec50 data for complexid = 50000963
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50393257(CHEMBL2151735)
Affinity DataEC50:  0nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse frontal cortex assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50393258(CHEMBL2151734)
Affinity DataEC50:  0nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse frontal cortex assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50376594(CHEMBL260120)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse frontal cortex assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50554766(CHEMBL4795492)
Affinity DataEC50:  0.0316nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50554766(CHEMBL4795492)
Affinity DataEC50:  0.0320nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50393258(CHEMBL2151734)
Affinity DataEC50:  0.287nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse spinal cord assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50393257(CHEMBL2151735)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse spinal cord assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50000507((R)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50376593(CHEMBL409225 | SB-0304)
Affinity DataEC50:  6.70nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse spinal cord assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50376593(CHEMBL409225 | SB-0304)
Affinity DataEC50:  567nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse frontal cortex assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Mu-type opioid receptor(MOUSE)
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50376594(CHEMBL260120)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at MOR/DOR in in NMRI mouse spinal cord assessed as reduction in spinal cord network activity by electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed