Compile Data Set for Download or QSAR
maximum 50k data
Found 52 of ki data for complexid = 220,50000168
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50111396(CHEMBL273636 | [[(S)-1-(4-Bromo-phenyl)-ethylamino...)
Affinity DataKi:  5.40nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50130937(Dexoxadrol | Dioxadrol)
Affinity DataKi:  19nMAssay Description:Inhibition of [3H]-U-69,593 binding to Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50130938(Etoxadrol)
Affinity DataKi:  22nMAssay Description:Binding affinity to NMDA receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50050704((R)-4-(3-Phosphono-propyl)-piperazine-2-carboxylic...)
Affinity DataKi:  41nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50044140(2-(2-Chloro-phenyl)-2-methylamino-cyclohexanone | ...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-MK801 from human forebrain GluN1/GluN2B expressed in HEK293 cells by at -70 mV holding potential by patch-clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50044140(2-(2-Chloro-phenyl)-2-methylamino-cyclohexanone | ...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-MK801 from rat brain GluN1/GluN2A expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419775(CHEMBL1950808)
Affinity DataKi:  210nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50004897((APV)2-Amino-5-phosphono-pentanoic acid | (R)-2-Am...)
Affinity DataKi:  280nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Affinity DataKi:  320nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164549((2R,3S)-1-(7-Bromo-phenanthrene-2-carbonyl)-pipera...)
Affinity DataKi:  320nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM81977(CAS_79055-68-8 | CB3371309 | D-AP5 | D-APV)
Affinity DataKi:  390nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50017226((R)-2-Amino-7-phosphono-heptanoic acid | 2-Amino-7...)
Affinity DataKi:  490nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  550nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164556((2R,3S)-1-((E)-3-Naphthalen-2-yl-acryloyl)-piperaz...)
Affinity DataKi:  840nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Affinity DataKi:  1.50E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164555((2R,3S)-1-(9,10-Dihydro-phenanthrene-2-carbonyl)-p...)
Affinity DataKi:  1.54E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419786(CHEMBL1950795)
Affinity DataKi:  3.00E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164548((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Affinity DataKi:  3.88E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164548((2R,3S)-1-(7-Bromo-9,10-dihydro-phenanthrene-2-car...)
Affinity DataKi:  3.90E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419787(CHEMBL1950794)
Affinity DataKi:  4.10E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50246910(CHEMBL4084540)
Affinity DataKi:  4.70E+3nMAssay Description:Antagonist activity at recombinant rat GluN1a/GluN2A expressed in Xenopus laevis oocytes assessed as inhibition of glycine/glutamate-mediated current...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419784(CHEMBL1950797)
Affinity DataKi:  5.10E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419778(CHEMBL1950803)
Affinity DataKi:  7.20E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419788(CHEMBL1950793)
Affinity DataKi:  7.40E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50364074(CHEMBL1950805)
Affinity DataKi:  7.40E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164545((2R,3S)-1-(9-Oxo-9H-fluorene-2-carbonyl)-piperazin...)
Affinity DataKi:  7.97E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164550((2R,3S)-1-(4'-Fluoro-biphenyl-4-carbonyl)-piperazi...)
Affinity DataKi:  8.78E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164551((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  9.60E+3nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164551((2R,3S)-1-(Naphthalene-2-carbonyl)-piperazine-2,3-...)
Affinity DataKi:  9.60E+3nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-(+)-MK-801 from phencyclidine binding site of NMDA receptor in human frontal cortex after 22 hrs by scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164543((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.05E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164543((2R,3R)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.05E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419776(CHEMBL1950806)
Affinity DataKi:  1.05E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164541((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Affinity DataKi:  1.12E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164541((2R,3S)-1-Phenanthren-2-ylmethyl-piperazine-2,3-di...)
Affinity DataKi:  1.12E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419777(CHEMBL1950804)
Affinity DataKi:  1.15E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164554((2R,3S)-1-[(E)-(3-Phenyl-acryloyl)]-piperazine-2,3...)
Affinity DataKi:  1.32E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164544((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.36E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164544((2R,3S)-1-(Biphenyl-4-sulfonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.36E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164553((2R,3S)-1-(Phenanthrene-3-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.42E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164552((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.57E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164552((2R,3S)-1-(Biphenyl-4-carbonyl)-piperazine-2,3-dic...)
Affinity DataKi:  1.58E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.76E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164540((2R,3S)-1-(Phenanthrene-2-carbonyl)-piperazine-2,3...)
Affinity DataKi:  1.76E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164553((2R,3S)-1-(Phenanthrene-3-carbonyl)-piperazine-2,3...)
Affinity DataKi:  2.20E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164542((2R,3S)-1-(2'-Bromo-biphenyl-4-carbonyl)-piperazin...)
Affinity DataKi:  4.29E+4nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419780(CHEMBL1950801)
Affinity DataKi:  9.93E+4nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419783(CHEMBL1950798)
Affinity DataKi: >1.00E+5nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50419779(CHEMBL1950802)
Affinity DataKi: >1.00E+5nMAssay Description:Antagonist activity at rat recombinant GluN1/GluN2A receptor expressed in Xenopus laevis oocytes assessed as inhibition of glutamate-induced response...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Rattus norvegicus (Rat))
University Walk

Curated by ChEMBL
LigandPNGBDBM50164547((2R,3S)-1-Benzoyl-piperazine-2,3-dicarboxylic acid...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibitory constant against (S)-glutamate and glycine evoked currents mediated by N-methyl-D-aspartate glutamate receptor NR1a/NR2A expressed in Xeno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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