Compile Data Set for Download or QSAR
Report error Found 56 of ki data for complexid = 50000206,50003479,50005181,50009808
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179395(CHEMBL14640)
Affinity DataKi:  0.891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138499(2-Phenethyl-4,5-dihydro-1H-imidazole | CHEMBL14210)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472306(CHEMBL93845)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138435(N-(12-Guanidino-dodecyl)-N-(1-phenethyl-piperidin-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50019848(CHEMBL10316 | Idazoxan | US8633208, Idazoxan | 4,5...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473129(Phenamazoline)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50121457(1-[3-(2,4-Dihydroxy-phenyl)-5-m-tolyl-4,5-dihydro-...)
Affinity DataKi:  50nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50121456(1-[3-(2,4-Dihydroxy-phenyl)-5-o-tolyl-4,5-dihydro-...)
Affinity DataKi:  80nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50474215(CHEMBL2092860)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179394(CHEMBL68608)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138436(N-(8-Guanidino-octyl)-N-(1-phenethyl-piperidin-4-y...)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091345(CHEMBL2092861)
Affinity DataKi:  145nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473618(CHEMBL337945)
Affinity DataKi:  182nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473198(CHEMBL13925)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473621(CHEMBL131775)
Affinity DataKi:  269nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50421578(CHEMBL13789)
Affinity DataKi:  302nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138434(N-(6-Guanidino-hexyl)-N-(1-phenethyl-piperidin-4-y...)
Affinity DataKi:  409nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138432(N-(2-Guanidino-ethyl)-N-(1-phenethyl-piperidin-4-y...)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50000214(CHEMBL337862)
Affinity DataKi:  813nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50472305(CHEMBL67706)
Affinity DataKi:  891nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091347(CHEMBL71429)
Affinity DataKi:  933nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  1.62E+3nMAssay Description:Binding affinity to imidazoline receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412250(CHEMBL128168)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50138433(N-(3-Guanidino-propyl)-N-(1-phenethyl-piperidin-4-...)
Affinity DataKi:  1.92E+3nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50179396(CHEMBL1907831)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50412260(CHEMBL273485)
Affinity DataKi:  2.69E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50008984(N-(1-Phenethyl-piperidin-4-yl)-N-phenyl-propionami...)
Affinity DataKi:  5.46E+3nMAssay Description:Displacement of [3H]2-BFI (1 nM) from imidazoline receptor I-2 in human brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50121455(1-[3-(2-Hydroxy-phenyl)-5-m-tolyl-4,5-dihydro-pyra...)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Bovine)
Sapienza University of Rome

Curated by ChEMBL
LigandPNGBDBM50045442(CHEMBL332286)
Affinity DataKi:  6.00E+3nMAssay Description:Inhibitory activity against Monoamine oxidase from Bovine brain mitochondriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50417354(CHEMBL396013)
Affinity DataKi:  7.24E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473620(CHEMBL131222)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473242(CHEMBL40287)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473240(CHEMBL40337)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473237(CHEMBL40393)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473241(CHEMBL288951)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473239(CHEMBL442156)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50070357(CHEMBL288139)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473238(CHEMBL40399)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]idazoxan from I2 imidazoline binding sites (I2Bs) of rabbit renal cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50091346(CHEMBL1907832)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 of rabbit kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A/B(Human)
University of Camerino

Curated by ChEMBL
LigandPNGBDBM50473619(CHEMBL130884)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of [3H]idazoxan from imidazoline receptor I-2 binding sites in rabbit kidney membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
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