Compile Data Set for Download or QSAR
Report error Found 17 of ki data for complexid = 50002812
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM30703(SMR000058526 | 2-[(4-tert-butyl-2,6-dimethyl-pheny...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50001922(Naphazoline | Albalon | Opcon | CHEMBL1706 | Nafaz...)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM96559(cid_10648 | Tetrahydrozoline hydrochloride | 2-(1,...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
LigandPNGBDBM50222199(CHEMBL157948)
Affinity DataKi:  500nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222135(CHEMBL347351)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222193(CHEBI:28611 | CHEMBL349584)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222194(CHEBI:28651 | CHEMBL348881)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222197(CHEBI:15944 | CHEMBL155870)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222196(CHEBI:46816 | CHEMBL155707)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222198(CHEBI:28658 | CHEMBL160579)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222195(Tetrahydropapaverine)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50027326(CHEMBL156383 | cid_440990 | (R)-norlaudanosoline |...)
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50027331(CHEMBL19068 | 1-[(3,4-dihydroxyphenyl)methyl]-1,2,...)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222134(CHEMBL160143)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed
LigandPNGBDBM50222200(CHEMBL160310)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of [3H]WB-4101 binding to alpha adrenergic receptor from rat cerebral cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2018
Entry Details Article
PubMed