Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50043404
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440622(CHEMBL2426556)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440621(CHEMBL2426554)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440620(CHEMBL2426552)
Affinity DataIC50: 1.63E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440619(CHEMBL2426555)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440627(CHEMBL2426553)
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440620(CHEMBL2426552)
Affinity DataIC50: 9.90E+4nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440624(CHEMBL2426550)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440625(CHEMBL2426549)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440626(CHEMBL2426548)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440622(CHEMBL2426556)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440619(CHEMBL2426555)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440621(CHEMBL2426554)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440627(CHEMBL2426553)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440623(CHEMBL2426551)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440624(CHEMBL2426550)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440625(CHEMBL2426549)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-oxoacyl-[acyl-carrier-protein] reductase(Plasmodium falciparum (isolate 3D7))
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440626(CHEMBL2426548)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum 3D7 FabG using acetoacetyl-CoA as substrate after 10 mins in presence of NADPHMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target3-hydroxyacyl-[acyl-carrier-protein] dehydratase(malaria parasite P. falciparum)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50440623(CHEMBL2426551)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant Plasmodium falciparum FabZ using crotonoyl-CoA as substrate after 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed