Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50009280
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526793(CHEMBL4562323)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526804(CHEMBL4553241)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2/cycE1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526792(CHEMBL4454044)
Affinity DataIC50: <5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526799(CHEMBL4440386)
Affinity DataIC50: <5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526798(CHEMBL4552441)
Affinity DataIC50: <5nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526793(CHEMBL4562323)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526804(CHEMBL4553241)
Affinity DataIC50:  14nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)
Affinity DataIC50:  14nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526788(CHEMBL4471850)
Affinity DataIC50:  18nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526801(CHEMBL4474655)
Affinity DataIC50: <20nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526790(CHEMBL4555799)
Affinity DataIC50: <20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526801(CHEMBL4474655)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK9 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526791(CHEMBL4465061)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526800(CHEMBL4533453)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526791(CHEMBL4465061)
Affinity DataIC50:  20nMAssay Description:Inhibition of CDK9 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)
Affinity DataIC50:  27nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)
Affinity DataIC50:  27nMAssay Description:Inhibition of CDK7 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  30nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526789(CHEMBL4459754)
Affinity DataIC50:  41nMAssay Description:Inhibition of CDK7/CycH/MAT1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526804(CHEMBL4553241)
Affinity DataIC50:  41nMAssay Description:Inhibition of CDK1 (unknown origin) by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5931(BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...)
Affinity DataIC50:  48nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526799(CHEMBL4440386)
Affinity DataIC50: <50nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526798(CHEMBL4552441)
Affinity DataIC50: <50nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526798(CHEMBL4552441)
Affinity DataIC50: <50nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526799(CHEMBL4440386)
Affinity DataIC50: <50nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526793(CHEMBL4562323)
Affinity DataIC50:  53nMAssay Description:Inhibition of CDK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5931(BMS-387072 | CHEMBL296468 | N-(5-{[(5-tert-butyl-1...)
Affinity DataIC50:  62nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  80nMAssay Description:Inhibition of CDK6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  90nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)
Affinity DataIC50:  97nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  100nMAssay Description:Inhibition of CDK4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526807(CHEMBL4467048 | US10870651, Compound 102)
Affinity DataIC50: <100nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526795(CHEMBL4450322)
Affinity DataIC50: >100nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  110nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526794(CHEMBL4303287 | US10787436, Compound I-18)
Affinity DataIC50:  134nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  170nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50:  170nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526806(CHEMBL4303279)
Affinity DataIC50:  194nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  200nMAssay Description:Inhibition of CDK5 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526790(CHEMBL4555799)
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526800(CHEMBL4533453)
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 7(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526802(CHEMBL4468921)
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK7 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526801(CHEMBL4474655)
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK2 (unknown origin) after 4 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Human)
Tianjin University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50526800(CHEMBL4533453)
Affinity DataIC50: >200nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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