Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50000096
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240523(CHEMBL4084630)
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240524(CHEMBL4079603)
Affinity DataIC50: 9.5nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240505(CHEMBL4077559)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240522(CHEMBL4067946)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240521(CHEMBL4095348)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240525(CHEMBL4070911)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240506(CHEMBL4103102)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240517(CHEMBL4066107)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240518(CHEMBL4103858)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50030448(CHEMBL269732 | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN ...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240516(CHEMBL4094558)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240519(CHEMBL4091778)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240511(CHEMBL4087653)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240508(CHEMBL4079773)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240526(CHEMBL4100390)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240515(CHEMBL4084186)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240507(CHEMBL4078827)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human FKBP12 measured after 30 mins by fluorescein labelled SLF tracer based fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240505(CHEMBL4077559)
Affinity DataIC50: 824nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240516(CHEMBL4094558)
Affinity DataIC50: 850nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240517(CHEMBL4066107)
Affinity DataIC50: 989nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240524(CHEMBL4079603)
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240518(CHEMBL4103858)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240525(CHEMBL4070911)
Affinity DataIC50: 1.11E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240521(CHEMBL4095348)
Affinity DataIC50: 1.29E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240523(CHEMBL4084630)
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240522(CHEMBL4067946)
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Amplyx Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50240506(CHEMBL4103102)
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at recombinant human N-terminal His6-tagged FKBP12 expressed in Escherichia coli assessed as inhibition of FK506 mediated FKBP12 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed