Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50000931
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010980(CHEMBL4089961)
Affinity DataKd:  0.0160nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010942(CHEMBL4077554)
Affinity DataKd:  0.0370nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50040717(CHEMBL4099729)
Affinity DataKd:  0.0933nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50054627(CHEMBL4070115)
Affinity DataKd:  2.40nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010980(CHEMBL4089961)
Affinity DataKd:  0.0160nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010971(CHEMBL4069112)
Affinity DataKd:  0.420nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50054627(CHEMBL4070115)
Affinity DataKd:  2.40nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010973(CHEMBL4091080)
Affinity DataKd:  1.60nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010974(CHEMBL4067866)
Affinity DataKd:  5.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010975(CHEMBL4075338)
Affinity DataKd:  0.170nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50040717(CHEMBL4099729)
Affinity DataKd:  0.0940nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010978(CHEMBL4077233)
Affinity DataKd:  0.710nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010963(CHEMBL4076226)
Affinity DataKd:  0.550nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010979(CHEMBL4072540)
Affinity DataKd:  2.40nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010943(CHEMBL4075701)
Affinity DataKd:  0.400nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50028301(CHEMBL4061407)
Affinity DataKd:  0.5nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010979(CHEMBL4072540)
Affinity DataKd:  2.40nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010963(CHEMBL4076226)
Affinity DataKd:  0.550nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010978(CHEMBL4077233)
Affinity DataKd:  0.708nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010975(CHEMBL4075338)
Affinity DataKd:  0.162nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010974(CHEMBL4067866)
Affinity DataKd:  5.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010973(CHEMBL4091080)
Affinity DataKd:  1.60nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010971(CHEMBL4069112)
Affinity DataKd:  0.417nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM165202(US9062043, Table 10, Compound 5 | US8168651, Compo...)
Affinity DataKd:  8.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKd:  0.562nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataKd:  0.560nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM165202(US9062043, Table 10, Compound 5 | US8168651, Compo...)
Affinity DataKd:  8.90nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010942(CHEMBL4077554)
Affinity DataKd:  0.0370nMAssay Description:Inhibition of ARC-1504 binding to CK2alpha (unknown origin) (1 to 335 residues) measured after 15 mins by fluorescence anisotropic methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlbumin(Bovine)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010963(CHEMBL4076226)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to bovine serum albumin by fluorescence anisotropy based methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlbumin(Bovine)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010943(CHEMBL4075701)
Affinity DataKd:  1.70E+3nMAssay Description:Binding affinity to bovine serum albumin by fluorescence anisotropy based methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010942(CHEMBL4077554)
Affinity DataIC50: 4nMAssay Description:Inhibition of CK2alpha (unknown origin) (1 to 335 residues) using 5-TAMRA-RADDSDDDDD as substrate after 30 mins by fluorescence imaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of CK2alpha (unknown origin) (1 to 335 residues) using 5-TAMRA-RADDSDDDDD as substrate after 30 mins by fluorescence imaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCasein kinase II subunit alpha(Human)
University of Tartu

Curated by ChEMBL
LigandPNGBDBM50010974(CHEMBL4067866)
Affinity DataIC50: 300nMAssay Description:Inhibition of CK2alpha (unknown origin) (1 to 335 residues) using 5-TAMRA-RADDSDDDDD as substrate after 30 mins by fluorescence imaging methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed