Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50003495
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50058715(CHEMBL64360 | EMD-96785 | N-(diaminomethylene)-2-m...)
Affinity DataIC50: 8nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471819(CHEMBL332433)
Affinity DataIC50: 13nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471814(CHEMBL126367)
Affinity DataIC50: 14nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471802(CHEMBL124274)
Affinity DataIC50: 16nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471801(CHEMBL331794)
Affinity DataIC50: 17nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471791(CHEMBL439605)
Affinity DataIC50: 19nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471796(CHEMBL124547)
Affinity DataIC50: 21nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471794(CHEMBL124044)
Affinity DataIC50: 24nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50234609(Cariporide | HOE-642)
Affinity DataIC50: 26nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471811(CHEMBL126060)
Affinity DataIC50: 27nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471823(CHEMBL341296)
Affinity DataIC50: 28nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471812(CHEMBL331630)
Affinity DataIC50: 28nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471815(CHEMBL123578)
Affinity DataIC50: 29nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471805(CHEMBL122142)
Affinity DataIC50: 30nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471808(CHEMBL333059)
Affinity DataIC50: 34nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471803(CHEMBL123859)
Affinity DataIC50: 36nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471804(CHEMBL421240)
Affinity DataIC50: 38nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471813(CHEMBL331457)
Affinity DataIC50: 40nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471807(CHEMBL125283)
Affinity DataIC50: 43nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471818(CHEMBL273539)
Affinity DataIC50: 44nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471816(CHEMBL125952)
Affinity DataIC50: 45nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471795(CHEMBL123160)
Affinity DataIC50: 45nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471790(CHEMBL333480)
Affinity DataIC50: 54nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471820(CHEMBL330935)
Affinity DataIC50: 56nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471799(CHEMBL124884)
Affinity DataIC50: 60nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471797(CHEMBL124762)
Affinity DataIC50: 60nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471809(CHEMBL333804)
Affinity DataIC50: 70nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471817(CHEMBL122853)
Affinity DataIC50: 93nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471792(CHEMBL340249)
Affinity DataIC50: 95nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471810(CHEMBL445376)
Affinity DataIC50: 96nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471821(CHEMBL121732)
Affinity DataIC50: 96nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471806(CHEMBL125951)
Affinity DataIC50: 116nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471793(CHEMBL121787)
Affinity DataIC50: 130nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471798(CHEMBL122238)
Affinity DataIC50: 360nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471824(CHEMBL124987)
Affinity DataIC50: 700nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471822(CHEMBL124826)
Affinity DataIC50: 790nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471800(CHEMBL333112)
Affinity DataIC50: 1.50E+3nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSodium/hydrogen exchanger 3(Rabbit)
Merck

Curated by ChEMBL
LigandPNGBDBM50471789(CHEMBL419609)
Affinity DataIC50: 2.20E+3nMAssay Description:Sodium/hydrogen exchanger antiport activity was measured using [22]Na+ uptake inhibition assay in acidified rabbit erythrocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed